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Record W2328677459 · doi:10.1021/om401050w

Electrophilic Aromatic Substitution Reactions of a Tungsten-Coordinated Phosphirenyl Triflate

2014· article· en· W2328677459 on OpenAlexaff
Arumugam Jayaraman, B.T. Sterenberg

Bibliographic record

VenueOrganometallics · 2014
Typearticle
Languageen
FieldChemistry
TopicOrganometallic Complex Synthesis and Catalysis
Canadian institutionsUniversity of Regina
Fundersnot available
KeywordsChemistryMedicinal chemistryElectrophilic aromatic substitutionSubstitution reactionTrifluoromethanesulfonateElectrophilic substitutionPyrroleStereochemistryOrganic chemistryCatalysis

Abstract

fetched live from OpenAlex

The phosphirenyl cation complex [W(CO) 5 {PC(Ph)C(Ph)}] + ( 2 ) is formed by chloride abstraction from the chlorophosphirene complex [W(CO) 5 {P(Cl)C(Ph)C(Ph)}] ( 1 ) with excess AlCl 3 . The phosphirenyl triflate complex [W(CO) 5 {P(OSO 2 CF 3 )C(Ph)C(Ph)}] ( 3 ) is formed by reaction of the chlorophosphirene complex with AgOSO 2 CF 3 and is in equilibrium with and typically reacts in the same fashion as the phosphirenyl cation. Reaction of 3 with diethylaniline or anisole leads to electrophilic aromatic substitution preferentially at the para position. Reaction with N, N -dimethyl- p -toluidine, in which the para position is blocked, leads to exclusive ortho substitution. The resulting 1,2-substituted arene can adopt a P,N bidentate coordination mode if a CO is removed from tungsten via photolysis. Compound 3 reacts with aromatic heterocycles thiophene, furan, and pyrrole, leading exclusively to substitution in the 2 position, with no evidence for P–S, P–O, or P–N bond formation. Reaction with indole led to substitution at the 3 position, also with no evidence for P–N bond formation. However, upon chromatographic purification, the substituted indole product decomposes into a disubstituted product, with W-coordinated phosphirenyl units at the 3 position and at N. Reaction with phenol and diphenyl amine led exclusively to P–O and P–N bond formation, with no evidence for aromatic substitution. Phosphine products can be removed via oxidation of W with I 2, followed by displacement with bipyridine. A computational study shows that coordination to W(CO) 5 greatly enhances electrophilicity at P in phosphenium ions, leading to the observed rapid electrophilic substitution reactions.

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

How this classification was reachedexpand

Full frame distilled prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. Learned from the 10,348 direct Codex labels and 10,348 direct Gemma labels. Candidate is the union of thresholded teacher heads; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels or direct frontier model labels.

metaresearch head score (Codex)0.000
metaresearch head score (Gemma)0.000
Version: codex-gemma-dda1882f352aValidation status: machine_predicted_unvalidated
Candidate categoriesMeta-epidemiology (narrow), Insufficient payload (model declined to judge)
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Bench or experimental · Consensus signal: Bench or experimental
GenreCandidate signal: Empirical · Consensus signal: Empirical
Teacher disagreement score0.105
Threshold uncertainty score1.000

Codex and Gemma teacher scores by category

CategoryCodexGemma
Metaresearch0.0000.000
Meta-epidemiology (narrow)0.0000.000
Meta-epidemiology (broad)0.0010.000
Bibliometrics0.0000.001
Science and technology studies0.0000.000
Scholarly communication0.0000.000
Open science0.0000.000
Research integrity0.0000.000
Insufficient payload (model declined to judge)0.0150.000

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.009
GPT teacher head0.201
Teacher spread0.192 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it

Classification

machine, unvalidated

Machine predicted; a candidate call from one teacher head, not a consensus.

Study designBench or experimental
Domainnot available
GenreEmpirical

How this classification was reached, model by model and score by score, is at the end of the page under "How this classification was reached".

Quick stats

Citations10
Published2014
Admission routes1
Has abstractyes

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