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Record W2802246087 · doi:10.1002/ejic.201800455

Metal Coordination to Unsymmetric 1,<i>n′</i>‐Disubstituted Ferrocene Histidine Peptides

2018· article· en· W2802246087 on OpenAlexafffund
Annaleizle Ferranco, Keija Sun, Theodore Udaipaul, Heinz‐Bernhard Kraatz

Bibliographic record

VenueEuropean Journal of Inorganic Chemistry · 2018
Typearticle
Languageen
FieldChemistry
TopicFerrocene Chemistry and Applications
Canadian institutionsThe Scarborough HospitalUniversity of Toronto
FundersNatural Sciences and Engineering Research Council of Canada
KeywordsChemistryFerroceneMetalImidazoleLigand (biochemistry)Coordination complexPeptideStereochemistryHistidineMetal ions in aqueous solutionChirality (physics)ConjugateMedicinal chemistryCombinatorial chemistryOrganic chemistryReceptorElectrochemistry

Abstract

fetched live from OpenAlex

In this study, the coordination chemistry of unsymmetrical 1, n ′‐substituted ferrocene (Fc) peptide conjugates is explored, where the peptide substituents are two different histidine‐containing peptides. The resulting Fc‐conjugates serve as ligands for the formation of metal complexes, with the intention to generate complexes that possess a labile coordination site. The following Fc[CO‐His(Trt)‐OMe][COOMe] ( 1 ), Fc[CO‐His(Trt)‐Gly‐OMe][CO‐Gly‐OMe] ( 2 ), Fc[CO‐His(Trt)‐His(Trt)‐OMe][CO‐His(Trt)‐OMe] ( 3 ), and Fc[CO‐His(Trt)‐Gly‐His(Trt)‐OMe][CO‐Gly‐His(Trt)‐OMe] ( 4 ) were synthesized and characterized. Each compound forms discrete complexes with metal divalent metal ions Zn 2+ , Co 2+ and Cd 2+ , where a single metal ion is complexed by the metallo‐ligand, as was confirmed spectroscopically. The redox properties of the Fc group are influenced by metal coordination to the peptide substituents and anodic shifts occur upon the addition of metal ions. These follow the order Zn 2+ &gt; Cd 2+ &gt; Co 2+ . NMR experiments indicated imidazole rings are the site of metal coordination. Fc‐peptide conjugates display a switchable axial chirality that is dependent on metal complexation.

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

How this classification was reachedexpand

Full frame distilled prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. Learned from the 10,348 direct Codex labels and 10,348 direct Gemma labels. Candidate is the union of thresholded teacher heads; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels or direct frontier model labels.

metaresearch head score (Codex)0.000
metaresearch head score (Gemma)0.001
Version: codex-gemma-dda1882f352aValidation status: machine_predicted_unvalidated
Candidate categoriesMeta-epidemiology (narrow), Insufficient payload (model declined to judge)
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Bench or experimental · Consensus signal: Bench or experimental
GenreCandidate signal: Empirical · Consensus signal: Empirical
Teacher disagreement score0.082
Threshold uncertainty score1.000

Codex and Gemma teacher scores by category

CategoryCodexGemma
Metaresearch0.0000.001
Meta-epidemiology (narrow)0.0000.000
Meta-epidemiology (broad)0.0000.000
Bibliometrics0.0000.001
Science and technology studies0.0000.000
Scholarly communication0.0000.000
Open science0.0010.000
Research integrity0.0000.000
Insufficient payload (model declined to judge)0.0030.000

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.014
GPT teacher head0.231
Teacher spread0.217 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it

Classification

machine, unvalidated

Machine predicted; a candidate call from one teacher head, not a consensus.

Study designBench or experimental
Domainnot available
GenreEmpirical

How this classification was reached, model by model and score by score, is at the end of the page under "How this classification was reached".

Quick stats

Citations6
Published2018
Admission routes2
Has abstractyes

Explore more

Same venueEuropean Journal of Inorganic ChemistrySame topicFerrocene Chemistry and ApplicationsFrench-language works237,207