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Record W2883672390 · doi:10.1111/bph.14453

Endocannabinoid regulation of homeostatic feeding and stress‐induced alterations in food intake in male rats

2018· article· en· W2883672390 on OpenAlexafffund
Martin A. Sticht, David J Lau, Catherine M. Keenan, Jean‐Baptiste Cavin, Maria Morena, Venkata Kiran Vemuri, Alexandros Makriyannis, Benjamin F. Cravatt, Keith A. Sharkey, Matthew N. Hill

Bibliographic record

VenueBritish Journal of Pharmacology · 2018
Typearticle
Languageen
FieldMedicine
TopicCannabis and Cannabinoid Research
Canadian institutionsHotchkiss Brain InstituteUniversity of Calgary
FundersCanadian Institutes of Health ResearchNational Institutes of Health
KeywordsEndocannabinoid systemMonoacylglycerol lipaseAnandamideEndocrinologyFatty acid amide hydrolaseInternal medicineCannabinoid receptorRimonabantHomeostasisCannabinoidAnorecticPharmacologyMedicineAntagonistReceptorFood intake

Abstract

fetched live from OpenAlex

Background and Purpose Stress is known to reduce food intake. Many aspects of the stress response and feeding are regulated by the endocannabinoid system, but the roles of anandamide (AEA) and 2‐arachidonoyl glycerol (2‐AG) in stress‐induced anorexia are unclear. Experimental Approach Effects of acute restraint stress on endocannabinoids were investigated in male Sprague–Dawley rats. Systemic and central pharmacological inhibition of fatty acid amide hydrolase (FAAH) or monoacylglycerol lipase (MAGL) was used to assess the effects of elevated AEA and 2‐AG on homeostatic feeding and on food consumption after stress. Animals were pretreated with the FAAH inhibitor, PF‐04457845, or the MAGL inhibitor, MJN110, before 2 h acute restraint stress or 2 h homecage period without food. Key Results Restraint stress decreased hypothalamic and circulating AEA, with no effect in the gastrointestinal tract, while 2‐AG content in the jejunum (but not duodenum) was reduced. PF‐04457845 (30 μg), given i.c.v., attenuated stress‐induced anorexia via CB 1 receptors, but reduced homeostatic feeding in unstressed animals through an unknown mechanism. On the other hand, systemic administration of MJN110 (10 mg·kg −1 ) reduced feeding, regardless of stress or feeding status and inhibited basal intestinal transit in unstressed rats. The ability of MAGL inhibition to reduce feeding in combination with stress was independent of CB 1 receptor signalling in the gut as the peripherally restricted CB 1 receptor antagonist, AM6545 did not block this effect. Conclusions and Implications Our data reveal diverse roles for 2‐AG and AEA in homeostatic feeding and changes in energy intake following stress. Linked Articles This article is part of a themed section on 8 th European Workshop on Cannabinoid Research. To view the other articles in this section visit http://onlinelibrary.wiley.com/doi/10.1111/bph.v176.10/issuetoc

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

How this classification was reachedexpand

Full frame machine prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. The Gemma side is a direct model label for every work in the frame, read from the title-only record. The Codex side is a classifier learned from the 10,348 direct Codex labels and calibrated to design-weighted sample rates; fields without enough sample support carry no Codex call. Candidate is the union of the two sides; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels.

metaresearch head score (Codex)0.000
metaresearch head score (Gemma)0.000
Version: metacan-v3-hybrid-931329e0061cValidation status: machine_predicted_unvalidated
Candidate categoriesnone
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Bench or experimental · Consensus signal: Bench or experimental
GenreCandidate signal: Empirical · Consensus signal: Empirical
Teacher disagreement score0.003
Threshold uncertainty score0.011

Distilled classifier scores by category (both heads)

CategoryCodexGemma
Metaresearch0.0000.000
Meta-epidemiology (narrow)0.0020.001
Meta-epidemiology (broad)0.0010.001
Bibliometrics0.0010.000
Science and technology studies0.0010.001
Scholarly communication0.0000.001
Open science0.0010.000
Research integrity0.0010.001
Insufficient payload (model declined to judge)0.0030.001

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.023
GPT teacher head0.326
Teacher spread0.304 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it

Classification

machine, unvalidated

Machine predicted; a candidate call from one source (direct Gemma or distilled Codex), not a consensus.

The models applied no category: nothing in the taxonomy fit this work.
Study designBench or experimental
Domainnot available
GenreEmpirical

How this classification was reached, model by model and score by score, is at the end of the page under "How this classification was reached".

Quick stats

Citations27
Published2018
Admission routes2
Has abstractyes

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