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Record W2949859869 · doi:10.1055/s-2000-6345

Allenylketenes: Versatile Substrates in Nucleophilic, Electrophilic, and Cycloaddition Reactions

2000· article· en· W2949859869 on OpenAlex

Why this work is in the frame

A frame that forgets how it found something cannot be audited. These are the routes that admitted this work.

affAt least one author lists a Canadian institution in the pinned OpenAlex snapshot.
fundA Canadian funder is recorded on the work.

Bibliographic record

VenueSynthesis · 2000
Typearticle
Languageen
FieldChemistry
TopicOrganic Chemistry Cycloaddition Reactions
Canadian institutionsUniversity of Toronto
FundersNatural Sciences and Engineering Research Council of Canada
KeywordsChemistryElectrophileCycloadditionNucleophileTrimethylsilylMedicinal chemistryBenzaldehydeAnilineKeteneStereochemistryOrganic chemistryCatalysis

Abstract

fetched live from OpenAlex

4-Methylene-2-trimethylsilyl-3-phenylcyclobutenones 3 are obtained from the corresponding cyclobutenedione 7 by Tebbe and Peterson methylenation reactions, and upon photolysis give 3-phenyl substituted allenylketenes R1CH=C=C(Ph)C(SiMe3)=C=O 4. These are more reactive in ring closure back to 3 than are the 3-trimethylsilyl analogs 1, as predicted on the basis of molecular orbital calculations. Reactions of allenylketenes 1 and 4 include addition of H2O followed by cyclization to form butenolides 13, addition of aniline to give allenyl carboxamide 14 and lactam 15, addition of CF3CO2H to form allenyl carboxylic acid 17, addition of Br2 in a 1,4-fashion to give penta-2,4-dienoic acid derivatives 18, and reaction with m-chloroperbenzoic acid to give the unique allenyl acylsilane 23. [4 + 1]-Cycloaddition reactions of 1 and 4 with Me3SiCHN2 give methylenecyclopentenones 24 and 25 while acetaldehyde undergoes BF3 · OEt2 catalyzed [2 + 2] cycloadditions forming β-lactones. [4 + 2] Cycloadditions occur with benzaldehyde to form the highly crowded exomethylene pentenolactone 29, and with TCNE forming methylenecyclohexenones 31.

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

Full frame distilled prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. Learned from the 10,348 direct Codex labels and 10,348 direct Gemma labels. Candidate is the union of thresholded teacher heads; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels or direct frontier model labels.

metaresearch head score (Codex)0.000
metaresearch head score (Gemma)0.000
Version: codex-gemma-dda1882f352aValidation status: machine_predicted_unvalidated
Candidate categoriesMeta-epidemiology (narrow), Insufficient payload (model declined to judge)
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Bench or experimental · Consensus signal: Bench or experimental
GenreCandidate signal: Empirical · Consensus signal: Empirical
Teacher disagreement score0.088
Threshold uncertainty score1.000

Codex and Gemma teacher scores by category

CategoryCodexGemma
Metaresearch0.0000.000
Meta-epidemiology (narrow)0.0000.000
Meta-epidemiology (broad)0.0000.000
Bibliometrics0.0000.000
Science and technology studies0.0000.000
Scholarly communication0.0000.000
Open science0.0000.000
Research integrity0.0000.000
Insufficient payload (model declined to judge)0.0760.000

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.006
GPT teacher head0.196
Teacher spread0.191 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it