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Record W3168044485 · doi:10.1136/heartjnl-2021-bcs.230

BS32 The role of branched-chain keto acids in mediating insulin resistance in the failing heart

2021· article· en· W3168044485 on OpenAlexaff
Qutuba G. Karwi, Cory S. Wagg, Liyan Zhang, John R. Ussher, Gary D. Lopaschuk

Bibliographic record

Venuenot available
Typearticle
Languageen
FieldBiochemistry, Genetics and Molecular Biology
TopicCancer, Hypoxia, and Metabolism
Canadian institutionsUniversity of Alberta
Fundersnot available
KeywordsInternal medicineEndocrinologyInsulin resistanceInsulinMedicineProtein kinase BHeart failureBranched-chain amino acidAmino acidBiologyPhosphorylationBiochemistry

Abstract

fetched live from OpenAlex

Brief introduction: Perturbed branched-chain amino acids (BCAA) oxidation positively correlates with the severity of cardiac insulin resistance in heart failure. We previously demonstrated that cardiac-specific deletion of the BCAA oxidative enzyme mitochondrial branched-chain aminotransferase (BCATm) increases cardiac BCAA levels and decreases branched-chain keto acids (BCKA) levels, enhances insulin-stimulated cardiac glucose oxidation rates. This increased cardiac insulin sensitivity is associated with an increase in the phosphorylation of protein kinase B (Akt) and activation of pyruvate dehydrogenase (PDH), the rate-limiting enzyme of glucose oxidation. However, whether it is the accumulation of BCAA or BCKA that is critical in mediating cardiac insulin resistance is unknown. How perturbed BCAA oxidation may mediate cardiac insulin resistance in heart failure is also unknown. Explanation of basic Methods To address these questions, we first examined the effects of selectively enhancing cardiac BCKA levels on cardiac insulin-stimulated glucose oxidation. We perfused isolated working mice hearts (male and female C57BL/6N, n=8-10) with high levels of BCKA (α-keto-isocaproate 80 μM, α-keto-β-methylvalorate 100μM, α-keto-isovalerate 70 μM), levels that can be seen in diabetes and obesity. Results High levels of BCKA completely blunted insulin-stimulated glucose oxidation rates and increased fatty acid oxidation rates. We also found that BCKA abolished insulin-stimulated mitochondrial Akt, an effect that was associated with PDH deactivation. We next determined the potential protective effect of reducing cardiac BCKA levels in the failing heart. We randomized WTCre+/+ and cardiac-specific BCATm-/- mice (male, 25-30g, n=6-8) to undergo either sham surgery or transverse aortic constriction surgery to induce heart failure. Five weeks post-surgery, there was a marked increase in insulin-stimulated glucose oxidation rates in the BCATm-/- failing hearts compared to the WTCre+/+ failing hearts, with no significant effect on glycolysis rates. Enhanced cardiac insulin sensitivity was associated with a significant decrease in fatty acid oxidation rates in the BCATm-/- failing hearts compared to the WTCre+/+ failing hearts. This decrease in fatty acid oxidation in the BCATm-/- failing hearts was associated with a significant decrease in myocardial oxygen consumption rates. As a result, cardiac efficiency (cardiac work/myocardial oxygen consumption) was significantly increased in the BCATm-/- failing hearts compared to the WTCre+/+ failing hearts. Conclusions/implications We conclude that the accumulation of BCKA, and not BCAA, is a major contributor to cardiac insulin resistance via abrogating mitochondrial translocation of Akt. Targeting BCKA may represent a potential therapeutic approach to improve cardiac insulin-stimulated glucose oxidation in the setting of heart failure, obesity and diabetes. Conflict of Interest None

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

How this classification was reachedexpand

Full frame machine prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. The Gemma side is a direct model label for every work in the frame, read from the title-only record. The Codex side is a classifier learned from the 10,348 direct Codex labels and calibrated to design-weighted sample rates; fields without enough sample support carry no Codex call. Candidate is the union of the two sides; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels.

metaresearch head score (Codex)0.000
metaresearch head score (Gemma)0.000
Version: metacan-v3-hybrid-931329e0061cValidation status: machine_predicted_unvalidated
Candidate categoriesnone
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Bench or experimental · Consensus signal: Bench or experimental
GenreCandidate signal: Empirical · Consensus signal: Empirical
Teacher disagreement score0.010
Threshold uncertainty score0.034

Distilled classifier scores by category (both heads)

CategoryCodexGemma
Metaresearch0.0000.000
Meta-epidemiology (narrow)0.0000.000
Meta-epidemiology (broad)0.0000.000
Bibliometrics0.0000.000
Science and technology studies0.0000.000
Scholarly communication0.0000.000
Open science0.0000.000
Research integrity0.0010.001
Insufficient payload (model declined to judge)0.0100.002

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.006
GPT teacher head0.234
Teacher spread0.227 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it

Classification

machine, unvalidated

Machine predicted; a candidate call from one source (direct Gemma or distilled Codex), not a consensus.

The models applied no category: nothing in the taxonomy fit this work.
Study designBench or experimental
Domainnot available
GenreEmpirical

How this classification was reached, model by model and score by score, is at the end of the page under "How this classification was reached".

Quick stats

Citations0
Published2021
Admission routes1
Has abstractyes

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