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P982: EFFICACY AND SAFETY OF 40 MG VS 60 MG OF ONCE WEEKLY SELINEXOR IN COMBINATION WITH POMALIDOMIDE AND DEXAMETHASONE IN RELAPSED AND/OR REFRACTORY MULTIPLE MYELOMA (RRMM)

2023· article· en· W4386074681 on OpenAlexaff
Darrell White, Muhamed Baljević, Gary J. Schiller, Suzanne Lentzsch, Evgeni Chubar, Noa Lavi, Dane R. Van Domelen, Ohad S. Bentur, Sumit Madan

Bibliographic record

VenueHemaSphere · 2023
Typearticle
Languageen
FieldMedicine
TopicMultiple Myeloma Research and Treatments
Canadian institutionsDalhousie University
Fundersnot available
KeywordsPomalidomideLenalidomideDexamethasoneMedicineMultiple myelomaRefractory (planetary science)BortezomibInternal medicineGastroenterologyOncology

Abstract

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Topic: 14. Myeloma and other monoclonal gammopathies - Clinical Background: Selinexor is an oral exportin 1 inhibitor approved with low-dose dexamethasone + bortezomib for patients (pts) with previously treated multiple myeloma (MM). Prior studies have reported an overall response rate (ORR) of 28% and a median progression free survival (mPFS) of 3.7 months to pomalidomide + low dose dexamethasone (Pd) in pts with MM refractory to both bortezomib and lenalidomide. STOMP is an ongoing Phase 1b/2 study evaluating selinexor in various triplet/quadruplet combinations in pts with newly diagnosed and relapsed/refractory MM (NCT02343042). In the selinexor + Pd (SPd) arm of the STOMP study, selinexor was evaluated at doses of 60-80 mg twice weekly (BIW; weeks 1-3 only) or 40-100 mg once weekly (QW) in combination with pomalidomide 2-4 mg once daily (QD, days 1-21) and dexamethasone 40 mg weekly) in 28-day treatment cycles. Aims: To identify the optimal dose of SPd, two expansion cohorts, with selinexor 60 mg QW (SPd-60) or 40 mg QW (SPd-40), both with pomalidomide 4 mg QD, were enrolled in STOMP and XPORT-MM-028, a parallel study with similar objectives and eligibility criteria (NCT04414475). Methods: We analyzed data of pts with RRMM treated with SPd in the STOMP and XPORT-MM-028 studies. Efficacy and safety of the combination were analyzed and compared by dose. Results: As of Sept 6, 2022, 28 pts with a median of 2.0 prior treatment lines (mLOT) and 20 pts with 2.5 mLOT were enrolled in the SPd-40 cohort and SPd-60 cohort, respectively. Among pts treated with SPd-40 and SPd-60, 93% and 75% had MM refractory to a proteasome inhibitor (PI), 75% and 85% had MM refractory to an immunomodulatory drug (IMiD), and 43% and 20% had triple-class refractory MM refractory to an anti-CD38 monoclonal antibody (αCD38 mAb), a PI and an IMiD, respectively. Prior exposure to αCD38 mAbs was reported in 57% and 30% of pts in the SPd-40 and SPd-60 cohorts, respectively. Median duration of exposure in the SPd-40 vs SPd-60 cohorts was 28 vs 22 weeks. Numerically higher ORR and rate of pts with ≥very good partial response (VGPR) were observed for SPd-60 vs SPd-40 (ORR: 65% vs 50%; ≥VGPR: 30% vs 25%), but the PFS was numerically longer for SPd-40 vs SPd-60 (mPFS in months: not reached [95% CI, 6.5-NE] after median follow-up of 1 year vs 9.5 months [95% CI, 7.6-NE]; 9-month PFS probability: 0.59 [95% CI, 0.41-0.85] vs 0.52 [95% CI, 0.29-0.94]). Across both doses among pts previously treated with αCD38 mAbs (n=22), mPFS was 8.9 months (95% CI, 6.5-NE). For the 27 responders across both doses, median time to response was 1.0 month (95% CI, 1-2) and median duration of response was 21.8 months (95% CI, 8.6-NE). Common hematologic treatment-emergent adverse events (TEAEs) included (all grades: SPd-40 vs SPd-60) neutropenia (68% vs 75% with one case of grade 3 febrile neutropenia in each cohort), anemia (39% vs 65%) and thrombocytopenia (43% vs 45%). No high-grade hemorrhages were observed. Non-hematologic TEAEs were generally transient and reversible, including fatigue (43% vs 75%), nausea (32% vs 70%) and diarrhea (25% vs 35%). Summary/Conclusion: The all-oral combination of selinexor + Pd in pts with RRMM was effective and tolerable in these cohorts. Most TEAEs, including nausea, occurred at lower frequency in the 40 mg cohort. Although a higher 60 mg QW selinexor dose may be associated with a higher ORR, mPFS correlated with longer duration on treatment is numerically longer for pts treated with the 40 mg dose, suggesting that clinical benefit is optimized at the lower 40 mg dose. SPd is being further evaluated in the EMN29 Phase 3 study (NCT05028348). Keywords: Multiple myeloma, Clinical trial, relapsed/refractory, Therapy

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How this classification was reachedexpand

Full frame distilled prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. Learned from the 10,348 direct Codex labels and 10,348 direct Gemma labels. Candidate is the union of thresholded teacher heads; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels or direct frontier model labels.

metaresearch head score (Codex)0.000
metaresearch head score (Gemma)0.001
Version: codex-gemma-dda1882f352aValidation status: machine_predicted_unvalidated
Candidate categoriesnone
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Observational · Consensus signal: Observational
GenreCandidate signal: Empirical · Consensus signal: Empirical
Teacher disagreement score0.097
Threshold uncertainty score0.557

Codex and Gemma teacher scores by category

CategoryCodexGemma
Metaresearch0.0000.001
Meta-epidemiology (narrow)0.0000.000
Meta-epidemiology (broad)0.0010.000
Bibliometrics0.0000.001
Science and technology studies0.0000.000
Scholarly communication0.0000.000
Open science0.0000.000
Research integrity0.0000.000
Insufficient payload (model declined to judge)0.0000.000

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.029
GPT teacher head0.303
Teacher spread0.273 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it

Classification

machine, unvalidated

Machine predicted; a candidate call from one teacher head, not a consensus.

The models applied no category: nothing in the taxonomy fit this work.
Study designObservational
Domainnot available
GenreEmpirical

How this classification was reached, model by model and score by score, is at the end of the page under "How this classification was reached".

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Citations1
Published2023
Admission routes1
Has abstractyes

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