MétaCan
Menu
Back to cohort
Record W4386396167 · doi:10.26434/chemrxiv-2023-hfcm5

Transfer Learning Graph Representations of Molecules for pKa, 13C-NMR, and Solubility

2023· preprint· en· W4386396167 on OpenAlexafffund
Amer Marwan El Samman, Stefano De Castro, Brooke Morton, Stijn De Baerdemacker

Bibliographic record

VenueChemRxiv · 2023
Typepreprint
Languageen
FieldComputer Science
TopicComputational Drug Discovery Methods
Canadian institutionsUniversity of New Brunswick
FundersNatural Sciences and Engineering Research Council of CanadaCanada Research ChairsCanada Foundation for InnovationNew Brunswick Innovation Foundation
KeywordsMolecular graphEmbeddingGraphChemical shiftAtom (system on chip)Representation (politics)MoleculeComputer scienceConvolutional neural networkChemistryArtificial intelligenceTheoretical computer sciencePhysical chemistry

Abstract

fetched live from OpenAlex

We explore transfer learning models from a pre-trained graph convoluntional neural network representation of molecules, obtained from SchNet, 1 to predict 13 C-NMR, pKa, and logS sol- ubility. SchNet learns a graph representation of a molecule by associating each atom with an “embedding vector” and interacts the atom-embeddings with each other by leveraging graph- convolutional filters on their interatomic distances. We pre-trained SchNet on molecular energy and demonstrate that the pre-trained atomistic embeddings can then be used as a transferable representation for a wide array of properties. On the one hand, for atomic properties such as micro-pK1 and 13 C-NMR, we investigate two models, one linear and one neural net, that inputs pre-trained atom-embeddings of a particular atom (e.g. carbon) and predicts a local property (e.g. 13 C-NMR). On the other hand, for molecular properties such as solubility, a size-extensive graph model is built using the embeddings of all atoms in the molecule as input. For all cases, qualitatively correct predictions are made with relatively little training data (<1000 training points), showcasing the ease with which pre-trained embeddings pick up on important chemical patterns. The proposed models successfully capture well-understood trends of pK1 and solu- bility. This study advances our understanding of current neural net graph representations and their capacity for transfer learning applications in chemistry.

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

How this classification was reachedexpand

Full frame distilled prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. Learned from the 10,348 direct Codex labels and 10,348 direct Gemma labels. Candidate is the union of thresholded teacher heads; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels or direct frontier model labels.

metaresearch head score (Codex)0.001
metaresearch head score (Gemma)0.000
Version: codex-gemma-dda1882f352aValidation status: machine_predicted_unvalidated
Candidate categoriesnone
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Simulation or modeling · Consensus signal: Simulation or modeling
GenreCandidate signal: Empirical · Consensus signal: none
Teacher disagreement score0.554
Threshold uncertainty score0.926

Codex and Gemma teacher scores by category

CategoryCodexGemma
Metaresearch0.0010.000
Meta-epidemiology (narrow)0.0000.000
Meta-epidemiology (broad)0.0000.000
Bibliometrics0.0000.000
Science and technology studies0.0000.000
Scholarly communication0.0000.000
Open science0.0010.001
Research integrity0.0000.000
Insufficient payload (model declined to judge)0.0000.000

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.070
GPT teacher head0.352
Teacher spread0.282 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it

Classification

machine, unvalidated

Machine predicted; a candidate call from one teacher head, not a consensus.

The models applied no category: nothing in the taxonomy fit this work.
Study designSimulation or modeling
Domainnot available
GenreEmpirical

How this classification was reached, model by model and score by score, is at the end of the page under "How this classification was reached".

Quick stats

Citations3
Published2023
Admission routes2
Has abstractyes

Explore more

Same venueChemRxivSame topicComputational Drug Discovery MethodsFrench-language works237,207