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Antitumor neodymium(III) complex with 1,10-phenanthroline and nitrate ligands: A comprehensive experimental-theoretical study, in silico pharmacokinetic and cytotoxic properties

2024· article· en· W4401841640 on OpenAlex

Why this work is in the frame

A frame that forgets how it found something cannot be audited. These are the routes that admitted this work.

fundA Canadian funder is recorded on the work.
no affNo Canadian affiliation: this work is invisible to an affiliation-only frame.
No Canadian affiliation. An affiliation-only frame, the usual design, would never have seen this work. It is one of the works that make the case for inverting the frame.

Bibliographic record

VenueJournal of Molecular Structure · 2024
Typearticle
Languageen
FieldMedicine
TopicMetal complexes synthesis and properties
Canadian institutionsnot available
FundersFundação para a Ciência e a TecnologiaFundação de Amparo à Pesquisa e ao Desenvolvimento Científico e Tecnológico do MaranhãoConselho Nacional de Desenvolvimento Científico e TecnológicoCoordenação de Aperfeiçoamento de Pessoal de Nível SuperiorUniversity of Alberta
KeywordsChemistryIn silicoNeodymiumPhenanthrolineNitrateCytotoxic T cellPharmacokineticsCombinatorial chemistryPharmacologyStereochemistryBiochemistryOrganic chemistryIn vitroGene

Abstract

fetched live from OpenAlex

Here we report the crystallization of the tris(nitrate-O,O')-bis(1,10-phenanthroline-N,N')-neodymium(III) complex by the slow solvent evaporation method. Structural, electronic, thermal, and vibrational properties have been explored and discussed. Additionally, all vibrational modes were carefully assigned, and geometric parameters and chemical reactivity indices were obtained from the results of density functional theory (DFT) calculations including solvation effects in dimethylformamide and water, as well as in vacuum. Moreover, a computational study using Hirshfeld surfaces identified and quantified the intermolecular interactions that stabilize the crystal lattice. X-ray powder diffraction results showed that the system has monoclinic symmetry with C2/c-space group and four monomers per unit cell (Z = 4). The thermoanalytical measurements revealed that the material has high thermal stability (≈ 300°C) and the experimental Raman and FT-IR spectroscopic data showed good correlation with the spectra calculated via DFT, where it was confirmed the influence of the solvents on the structure of the complex. Finally, cell viability assays showed that the neodymium(III) complex has cytotoxic activity and selectivity against MCF-7 (breast) and SiHa (cervical) cancer cells, with a potent biological effect. Complementary, a computational study of the pharmacokinetic profile was performed to support the experimental biological data via absorption, distribution, metabolism and elimination (ADME), and druglikeness.

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

Full frame distilled prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. Learned from the 10,348 direct Codex labels and 10,348 direct Gemma labels. Candidate is the union of thresholded teacher heads; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels or direct frontier model labels.

metaresearch head score (Codex)0.000
metaresearch head score (Gemma)0.000
Version: codex-gemma-dda1882f352aValidation status: machine_predicted_unvalidated
Candidate categoriesnone
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Bench or experimental · Consensus signal: Bench or experimental
GenreCandidate signal: Empirical · Consensus signal: Empirical
Teacher disagreement score0.026
Threshold uncertainty score0.633

Codex and Gemma teacher scores by category

CategoryCodexGemma
Metaresearch0.0000.000
Meta-epidemiology (narrow)0.0000.000
Meta-epidemiology (broad)0.0010.000
Bibliometrics0.0000.000
Science and technology studies0.0000.000
Scholarly communication0.0000.000
Open science0.0000.000
Research integrity0.0000.000
Insufficient payload (model declined to judge)0.0000.000

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.027
GPT teacher head0.294
Teacher spread0.267 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it