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Record W4417188403 · doi:10.1021/acsptsci.5c00647

Optimization of a Green Extraction Technique for Kratom (Ketum) Leaf Extract via Accelerated Solvent Extraction: Phytochemical Profiles, Cytotoxicity, and Antinociceptive Activity

2025· article· en· W4417188403 on OpenAlex
Nurul Najwa Rusmadi, Thiruventhan Karunakaran, Faiqah Ramli, Intan Safinar Ismail, Ramesh Kumar Santhanam, J. D. Yuvenesan Jagabalan, Mohamad Hafizi Abu Bakar, Azira Muhamad, Surash Ramanathan

Why this work is in the frame

A frame that forgets how it found something cannot be audited. These are the routes that admitted this work.

affAt least one author lists a Canadian institution in the pinned OpenAlex snapshot.

Bibliographic record

VenueACS Pharmacology & Translational Science · 2025
Typearticle
Languageen
FieldPharmacology, Toxicology and Pharmaceutics
TopicAlkaloids: synthesis and pharmacology
Canadian institutionsCentre for Drug Research and Development
FundersUniversiti Sains MalaysiaMinistry of Higher Education, Malaysia
KeywordsPhytochemicalCytotoxicityFlavonoidExtraction (chemistry)SolventPotencyEthanol

Abstract

fetched live from OpenAlex

Kratom ( Mitragyna speciosa Korth.) has gained increasing scientific interest for its potential in pain management and addiction treatment. This study employs a green chemistry approach to optimize the extraction of kratom leaves by using Accelerated Solvent Extraction (ASE) with an ethanol–water binary solvent system. The goal was to improve the yield and potency of key bioactive compounds, especially mitragynine. Optimization was performed using One-Factor-at-a-Time (OFAT) analysis and Response Surface Methodology (RSM) employing a Box-Behnken Design (BBD). The optimal extraction conditions were determined to be an 8 min extraction time, 60 °C temperature, and 40% ethanol concentration, which resulted in mitragynine content of 4.66%, total phenolic content of 212.69 GAE mg/g, and total flavonoid content of 126.13 QE mg/g. The safety profile of the optimized ASE kratom leaf extract was evaluated using MTT cytotoxicity assay, which revealed selective cytotoxicity against HepG2 liver cancer cells (IC 50 = 7.69 μg/mL), while showing no cytotoxicity toward HL-7702 normal liver cells (IC 50 > 200 μg/mL). Antinociceptive activity was tested in BALB/c albino mice using the hot-plate test, where the optimized ASE kratom leaf extract demonstrated analgesic effects at dosages of 100, 200, and 500 mg/kg. Phytochemical profiling combining NMR and UPLC-ESI-QTOF-MS/MS identified several known kratom constituents, including mitragynine and its congeners as well as bioactive flavonoids such as isoquercitrin and rutin. The optimized ASE method using a green ethanol–water system produces kratom extracts with promising safety and therapeutic potential, though further work is needed to refine and scale the approach for broader phytopharmaceutical use.

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

Full frame distilled prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. Learned from the 10,348 direct Codex labels and 10,348 direct Gemma labels. Candidate is the union of thresholded teacher heads; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels or direct frontier model labels.

metaresearch head score (Codex)0.002
metaresearch head score (Gemma)0.000
Version: codex-gemma-dda1882f352aValidation status: machine_predicted_unvalidated
Candidate categoriesMeta-epidemiology (narrow), Insufficient payload (model declined to judge)
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Bench or experimental · Consensus signal: Bench or experimental
GenreCandidate signal: Empirical · Consensus signal: Empirical
Teacher disagreement score0.215
Threshold uncertainty score1.000

Codex and Gemma teacher scores by category

CategoryCodexGemma
Metaresearch0.0020.000
Meta-epidemiology (narrow)0.0000.000
Meta-epidemiology (broad)0.0010.000
Bibliometrics0.0010.001
Science and technology studies0.0010.002
Scholarly communication0.0000.001
Open science0.0010.000
Research integrity0.0010.001
Insufficient payload (model declined to judge)0.0010.000

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.082
GPT teacher head0.447
Teacher spread0.364 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it