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Record W1919453433 · doi:10.1002/047084289x.rd263

1,5-Dilithiopentane

2001· reference-entry· en· W1919453433 on OpenAlexaff
P. Canonne, Paul Angers

Bibliographic record

VenueEncyclopedia of Reagents for Organic Synthesis · 2001
Typereference-entry
Languageen
FieldChemistry
TopicCoordination Chemistry and Organometallics
Canadian institutionsUniversité Laval
Fundersnot available
KeywordsReagentLithium (medication)ChemistryCyclohexaneEtherBifunctionalAnhydrousSolubilityPotentiometric titrationMetalHalideQuenching (fluorescence)Inorganic chemistryNuclear chemistryOrganic chemistryIonCatalysis

Abstract

fetched live from OpenAlex

[2223-58-7] C5H10Li2 (MW 84.02) InChI = 1S/C5H10.2Li/c1-3-5-4-2;;/h1-5H2;; InChIKey = QQDSVXYDUMVTSQ-UHFFFAOYSA-N (constructing block agent: transformations of carboxyl groups and metal halides into cyclohexane and metallacyclohexane synthetic intermediates, and α,ω-bifunctional compounds; in presence of CuI ion, the reagent is transformed into an organobiscuprate) Alternate Name: 1,5-pentanediyldilithium. Solubility: sol ether, THF, hydrocarbons. Form Supplied in: prepared in ether and used in solutions which usually range from 0.5 to 1.2 M. Analysis of Reagent Purity: titration;2 1H NMR α-CH2 signal δ −0.81 (t, J = 9 Hz);3 quenching with chlorotrimethylsilane;3, 4 GLC.5 Preparative Methods: was first prepared by direct reaction of 1,5-dibromopentane with Lithium metal at 0 °C in anhydrous ether.4, 8 This method was later improved by using lithium metal (4 equiv) containing 1% Na with 1,5-dichloropentane (1 equiv).5 The optimum procedure9 uses a 12.5% excess of lithium and maintains the temperature at 0 °C (eq 1). Yields up to 90% can be obtained by this method, which may also serve to prepare lower analogs. (1) The Barbier procedure, under ultrasonic irradiation, may also be used. In a particular case, 1,5-dibromopentane (2 equiv), methyl R(−)-2-methyloctanoate (1 equiv) and lithium (8 equiv) were reacted in THF at −25 °C for 25 min (see eq 3).10 1,5-Dilithiopentane can also be prepared by lithium–iodine exchange between t‐Butyllithium and 1,5-diiodopentane (eq 2).3 This method requires a temperature of −78 °C and 4 equiv of t-BuLi.2 The excess of reagent is important, as a stoichiometric amount leads to the corresponding cycloalkane almost quantitatively. (2) The procedure also generates, in excellent yields, lithio compounds from homoallylic-type iodides. Alkyl bromides and secondary iodides may also be used, but yields are lower. Handling, Storage, and Precautions: solutions are highly flammable; must be stored and handled in the absence of proton sources, carbon acids, and oxygen. Flasks and Schlenk tubes should be flushed with dry Ar or N2. At −20 °C, ether solutions have a useful life of one to four months.5, 6 At higher temperature (∼30 °C), organolithiums react readily with ethers.7

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

How this classification was reachedexpand

Full frame machine prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. The Gemma side is a direct model label for every work in the frame, read from the title-only record. The Codex side is a classifier learned from the 10,348 direct Codex labels and calibrated to design-weighted sample rates; fields without enough sample support carry no Codex call. Candidate is the union of the two sides; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels.

metaresearch head score (Codex)0.000
metaresearch head score (Gemma)0.000
Version: metacan-v3-hybrid-931329e0061cValidation status: machine_predicted_unvalidated
Candidate categoriesnone
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Not applicable · Consensus signal: none
GenreCandidate signal: Other · Consensus signal: none
Teacher disagreement score0.019
Threshold uncertainty score0.062

Distilled classifier scores by category (both heads)

CategoryCodexGemma
Metaresearch0.0000.000
Meta-epidemiology (narrow)0.0010.000
Meta-epidemiology (broad)0.0000.000
Bibliometrics0.0000.000
Science and technology studies0.0000.000
Scholarly communication0.0000.000
Open science0.0010.000
Research integrity0.0000.001
Insufficient payload (model declined to judge)0.0190.010

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.018
GPT teacher head0.251
Teacher spread0.233 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it

Classification

machine, unvalidated

Machine predicted; a candidate call from one source (direct Gemma or distilled Codex), not a consensus.

The models applied no category: nothing in the taxonomy fit this work.
Study designNot applicable
Domainnot available
GenreOther

How this classification was reached, model by model and score by score, is at the end of the page under "How this classification was reached".

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Citations0
Published2001
Admission routes1
Has abstractyes

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