MétaCan
Menu
Back to cohort
Record W1982475294 · doi:10.1021/op900004c

Polymorphic Crystallization and Transformation of the Anti-Viral/HIV Drug Stavudine

2009· article· en· W1982475294 on OpenAlex

Why this work is in the frame

A frame that forgets how it found something cannot be audited. These are the routes that admitted this work.

affAt least one author lists a Canadian institution in the pinned OpenAlex snapshot.

Bibliographic record

VenueOrganic Process Research & Development · 2009
Typearticle
Languageen
FieldMedicine
TopicHIV/AIDS drug development and treatment
Canadian institutionsWestern University
Fundersnot available
KeywordsStavudineHuman immunodeficiency virus (HIV)CrystallizationTransformation (genetics)VirologyDrugMedicinePharmacologyChemistryBiologyGeneticsAntiretroviral therapyViral loadOrganic chemistry

Abstract

fetched live from OpenAlex

The effect of supersaturation, nucleation temperature, cooling rate and solvent on the polymorphic crystallization of stavudine has been studied. Supersaturation is found to be the predominant controlling factor for the occurrence of polymorphs. When stavudine crystallizes from methanol or 2-propanol, form I nucleates preferentially at a low supersaturation level, whereas form II can be obtained at a high supersaturation level. When 1-butanol is used as solvent, apart from forms I and II, a newly found metastable form IV can crystallize out at a moderate supersaturation level. The relative stability of the above three polymorphs in decreasing order is: I > IV > II. In addition, the polymorphic transformation of stavudine in 2-propanol from form II to form I has been investigated by in situ Raman spectroscopy. The transformation rate is found to be accelerated significantly by increasing temperature and seeding with form I.

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

Full frame distilled prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. Learned from the 10,348 direct Codex labels and 10,348 direct Gemma labels. Candidate is the union of thresholded teacher heads; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels or direct frontier model labels.

metaresearch head score (Codex)0.001
metaresearch head score (Gemma)0.000
Version: codex-gemma-dda1882f352aValidation status: machine_predicted_unvalidated
Candidate categoriesnone
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Bench or experimental · Consensus signal: Bench or experimental
GenreCandidate signal: Empirical · Consensus signal: Empirical
Teacher disagreement score0.278
Threshold uncertainty score0.482

Codex and Gemma teacher scores by category

CategoryCodexGemma
Metaresearch0.0010.000
Meta-epidemiology (narrow)0.0000.000
Meta-epidemiology (broad)0.0000.000
Bibliometrics0.0000.001
Science and technology studies0.0000.000
Scholarly communication0.0000.000
Open science0.0000.000
Research integrity0.0000.000
Insufficient payload (model declined to judge)0.0000.000

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.020
GPT teacher head0.308
Teacher spread0.288 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it