MétaCan
Menu
Back to cohort
Record W1991513961 · doi:10.2174/1568013053586487

To be or not to be: Regulation of the Intrinsic Activity of GLUT4

2005· article· en· W1991513961 on OpenAlexafffund
Costin N. Antonescu, Farah S. L. Thong, Wenyan Niu, Eddy Karnieli, Amira Klip

Bibliographic record

VenueCurrent Medicinal Chemistry - Immunology Endocrine & Metabolic Agents · 2005
Typearticle
Languageen
FieldBiochemistry, Genetics and Molecular Biology
TopicMetabolism, Diabetes, and Cancer
Canadian institutionsHospital for Sick Children
FundersCanadian Institutes of Health Research
KeywordsGLUT4Glucose transporterGlucose uptakeInsulinImmunoelectron microscopyCellIntracellularBiologyTransporterCell biologyInternal medicineBiochemistryEndocrinologyMedicineGeneAntibody

Abstract

fetched live from OpenAlex

Insulin increases the rate of glucose uptake into muscle and fat cells. Numerous studies provide evidence that this is accomplished through an increase in the cell-surface amount of the facilitative glucose transporter GLUT4. Diverse techniques have been used to document a time-dependent gain in surface GLUT4, often in conjunction with a decrease in its intracellular content. These include subcellular fractionation coupled to immunoblotting, affinity photolabelling coupled to immunoprecipitation, and surface detection by immunofluorescence and immunoelectron microscopy. However, there are also abundant reports of a discrepancy between the extent of stimulation of the rate of glucose uptake by insulin and the increase in the amount of cell-surface transporters. One interpretation of this discrepancy is that insulin regulates the intrinsic activity of GLUT4 in addition to recruiting transporters to the cell surface. Several interpretations of this discrepancy can be offered, based on the experimental techniques used to measure glucose uptake and cell-surface GLUT4. Here we discuss the methods used to quantify these observations. Subsequently, we inspect the studies that have measured the insulin-stimulated increase in cell-surface GLUT4 concurrently with glucose uptake, in order to determine if there is realistic evidence to support the hypothesis that insulin regulates GLUT4 intrinsic activity. We conclude that in spite of various possible explanations for the discrepancy between the stimulation of glucose uptake and that of cell surface GLUT4, there is solid evidence to suggest that insulin increases the intrinsic activity of GLUT4. Keywords: insulin, glucose transporters (gluts), expression, translocation, plasma membrane (pm)

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

How this classification was reachedexpand

Full frame distilled prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. Learned from the 10,348 direct Codex labels and 10,348 direct Gemma labels. Candidate is the union of thresholded teacher heads; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels or direct frontier model labels.

metaresearch head score (Codex)0.000
metaresearch head score (Gemma)0.001
Version: codex-gemma-dda1882f352aValidation status: machine_predicted_unvalidated
Candidate categoriesnone
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Bench or experimental · Consensus signal: Bench or experimental
GenreCandidate signal: Empirical · Consensus signal: Empirical
Teacher disagreement score0.393
Threshold uncertainty score0.955

Codex and Gemma teacher scores by category

CategoryCodexGemma
Metaresearch0.0000.001
Meta-epidemiology (narrow)0.0000.000
Meta-epidemiology (broad)0.0010.000
Bibliometrics0.0000.000
Science and technology studies0.0000.000
Scholarly communication0.0000.000
Open science0.0010.000
Research integrity0.0000.000
Insufficient payload (model declined to judge)0.0000.000

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.031
GPT teacher head0.321
Teacher spread0.290 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it

Classification

machine, unvalidated

Machine predicted; a candidate call from one teacher head, not a consensus.

The models applied no category: nothing in the taxonomy fit this work.
Study designBench or experimental
Domainnot available
GenreEmpirical

How this classification was reached, model by model and score by score, is at the end of the page under "How this classification was reached".

Quick stats

Citations14
Published2005
Admission routes2
Has abstractyes

Explore more

Same venueCurrent Medicinal Chemistry - Immunology Endocrine & Metabolic AgentsSame topicMetabolism, Diabetes, and CancerFrench-language works237,207