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Record W2016017164 · doi:10.1021/ja805801j

Enzyme-like Acceleration for the Hydrolysis of a DNA Model Promoted by a Dinuclear Zn(II) Catalyst in Dilute Aqueous Ethanol

2008· article· en· W2016017164 on OpenAlexaff
C. Tony Liu, Alexei A. Neverov, R. S. Brown

Bibliographic record

VenueJournal of the American Chemical Society · 2008
Typearticle
Languageen
FieldBiochemistry, Genetics and Molecular Biology
TopicDNA and Nucleic Acid Chemistry
Canadian institutionsQueen's University
Fundersnot available
KeywordsChemistryCatalysisEthanolReaction rate constantAqueous solutionHydrolysisPhosphoric acidDissociation constantInorganic chemistryAlcoholKineticsSolventNuclear chemistryMedicinal chemistryOrganic chemistry

Abstract

fetched live from OpenAlex

The rates and products of cleavage of methyl (2-chloro-4-nitrophenyl) phosphate (2) promoted by a dinuclear Zn(II) complex (3) of 1,3-bis-N,N'(1,5,9-triazacyclododecyl)propane along with 1 equiv of ethoxide were investigated in ethanol solution containing small amounts of water (8 mM <or= [H2O] <or= 2.1 M) at 25 degreesC and sspH 7.9. The kinetics of decomposition of 5 x 10(-5) M 2 in the presence of varying [3] (0.03 mM <or= [3] <or= 0.12 mM) in ethanol containing 28 mM water show very strong saturation binding which is analyzed to give fitted values for the complex dissociation constant (Kd) and maximum catalytic rate constant (kcatmax) of 3.2 x 10(-8) M and 1.47 x 10(-3) s(-1). Product analysis indicates that the reaction in ethanol containing 28 mM and 2.1 M water produces 46% and 93% of the hydrolysis product (methyl phosphoric acid), with the remainder being ethanolysis product (ethyl methyl phosphate). Analysis of the kinetics of the reaction at 28 mM water indicates that second order rate constant for the catalytic reaction, given as kcatmax/Kd, is 4.6 x 104 M(-1) s(-1), is a factor of 8.4 x 10(10) larger than the second order rate constant (k2EtO) for the ethoxide promoted reaction of 2 in ethanol (5.5 +/- 0.3) x 10(-7) M(-1) s(-1). A more detailed analysis that considers the relative acidities of water and ethanol in ethanol solvent indicates that at sspH 7.9, the ethanolysis is accelerated by 2.3 x 10(14) times relative to the computed ethoxide reaction at that sspH, while the hydrolysis is accelerated by >or=1.6 x 10(17) times relative to the background hydroxide reaction, suggesting that complex 3 promotes the hydrolysis at least 1000 times more effectively than ethanolysis.

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

How this classification was reachedexpand

Full frame distilled prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. Learned from the 10,348 direct Codex labels and 10,348 direct Gemma labels. Candidate is the union of thresholded teacher heads; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels or direct frontier model labels.

metaresearch head score (Codex)0.000
metaresearch head score (Gemma)0.000
Version: codex-gemma-dda1882f352aValidation status: machine_predicted_unvalidated
Candidate categoriesnone
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Bench or experimental · Consensus signal: Bench or experimental
GenreCandidate signal: Empirical · Consensus signal: Empirical
Teacher disagreement score0.019
Threshold uncertainty score0.345

Codex and Gemma teacher scores by category

CategoryCodexGemma
Metaresearch0.0000.000
Meta-epidemiology (narrow)0.0000.000
Meta-epidemiology (broad)0.0000.001
Bibliometrics0.0000.000
Science and technology studies0.0000.000
Scholarly communication0.0000.000
Open science0.0010.000
Research integrity0.0000.000
Insufficient payload (model declined to judge)0.0000.000

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.010
GPT teacher head0.232
Teacher spread0.222 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it

Classification

machine, unvalidated

Machine predicted; a candidate call from one teacher head, not a consensus.

The models applied no category: nothing in the taxonomy fit this work.
Study designBench or experimental
Domainnot available
GenreEmpirical

How this classification was reached, model by model and score by score, is at the end of the page under "How this classification was reached".

Quick stats

Citations29
Published2008
Admission routes1
Has abstractyes

Explore more

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