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Record W2046828673 · doi:10.1139/v02-176

L'échelle p<i>K</i><sub>HB</sub> de basicité de liaison hydrogène des amines tertiaires aliphatiques

2002· article· en· W2046828673 on OpenAlex

Why this work is in the frame

A frame that forgets how it found something cannot be audited. These are the routes that admitted this work.

venuePublished in a venue whose home country is Canada.
no affNo Canadian affiliation: this work is invisible to an affiliation-only frame.
No Canadian affiliation. An affiliation-only frame, the usual design, would never have seen this work. It is one of the works that make the case for inverting the frame.

Bibliographic record

VenueCanadian Journal of Chemistry · 2002
Typearticle
Languageen
FieldChemistry
TopicMolecular Spectroscopy and Structure
Canadian institutionsnot available
Fundersnot available
KeywordsChemistrySteric effectsLone pairHydrogen bondMedicinal chemistryNitrogenBenzonitrilePolar effectInfrared spectroscopyAcceptorStereochemistryOrganic chemistryMolecule

Abstract

fetched live from OpenAlex

The hydrogen bond acceptor strength of 40 tertiary amines has been measured by Fourier transform – infrared (FTIR) spectrometry from their 1:1 complexation constant towards 4-fluorophenol in CCl 4 at 25°C (the pK HB scale). Also measured was the frequency shift, Δν(OH), of the ν(OH) band of methanol hydrogen-bonded to these amines. The comparison of the thermodynamic hydrogen bond basicity scale, pK HB , with the spectroscopic one, Δν(OH), and with the Brønsted pK a scale, points to the great sensitivity of pK HB to steric effects. The pK HB scale of tertiary amines extends from 2.71 for quinuclidine to –0.34 for N,N-diisopropyl-3-pentylamine. The main factors governing this important variation (17 kJ·mol –1 on the Gibbs energy scale) are the electron-withdrawing inductive effect and various kinds of steric effects (e.g., opening of the CNC angles and hindrance to OH fixation on the nitrogen lone pair). Infrared (IR) spectra show the attachment of 4-fluorophenol to the nitrile nitrogen of Me 2 NCH 2 C[Formula: see text]N and Me 2 NCH 2 CH 2 C[Formula: see text]N, to the oxygen of N-methylmorpholine, and to the π electrons of (HC[Formula: see text]CCH 2 ) 3 N and (PhCH 2 ) 3 N, in addition to the attachment to the amino nitrogen. In (PhCH 2 ) 3 N, the electron-withdrawing effect of the three benzyl substituents and, mainly, the very important congestion of the nitrogen lone pair reduce the nitrogen hydrogen-bond basicity almost to nothing, so that tribenzylamine, a nitrogen Brønsted base, turns to a π base in hydrogen bonding. From this example, the large differences between the pK HB and pK a scales of organic bases are emphasized.Key words: basicity, hydrogen bonding, tertiary amines, pK HB scale.

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

Full frame distilled prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. Learned from the 10,348 direct Codex labels and 10,348 direct Gemma labels. Candidate is the union of thresholded teacher heads; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels or direct frontier model labels.

metaresearch head score (Codex)0.000
metaresearch head score (Gemma)0.000
Version: codex-gemma-dda1882f352aValidation status: machine_predicted_unvalidated
Candidate categoriesMeta-epidemiology (narrow), Insufficient payload (model declined to judge)
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Bench or experimental · Consensus signal: Bench or experimental
GenreCandidate signal: Empirical · Consensus signal: Empirical
Teacher disagreement score0.018
Threshold uncertainty score1.000

Codex and Gemma teacher scores by category

CategoryCodexGemma
Metaresearch0.0000.000
Meta-epidemiology (narrow)0.0000.000
Meta-epidemiology (broad)0.0000.000
Bibliometrics0.0000.000
Science and technology studies0.0000.000
Scholarly communication0.0000.000
Open science0.0000.000
Research integrity0.0000.001
Insufficient payload (model declined to judge)0.0020.000

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.006
GPT teacher head0.198
Teacher spread0.192 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it