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Record W2070213303 · doi:10.2202/1553-3840.1283

Optimized St. John's Wort (Hypericum perforatum L.) Germplasm Lines Exert Cytotoxicity in HT-29 Colon Cancer Cells via Downregulation of NF-?B

2010· article· en· W2070213303 on OpenAlex

Why this work is in the frame

A frame that forgets how it found something cannot be audited. These are the routes that admitted this work.

affAt least one author lists a Canadian institution in the pinned OpenAlex snapshot.
aboutThe title or abstract carries a Canadian signal from the geographic lexicon.

Bibliographic record

VenueJournal of Complementary and Integrative Medicine · 2010
Typearticle
Languageen
FieldBiochemistry, Genetics and Molecular Biology
TopicBiological Activity of Diterpenoids and Biflavonoids
Canadian institutionsUniversity of WindsorUniversity of British Columbia, Okanagan CampusUniversity of British ColumbiaUniversity of Guelph
Fundersnot available
KeywordsHypericinHypericum perforatumHyperforinPharmacologyHypericumDownregulation and upregulationTumor necrosis factor alphaCancer cellCytotoxicityMedicineTraditional medicineCancerChemistryBiochemistryImmunologyIn vitroInternal medicine

Abstract

fetched live from OpenAlex

Extracts of two germplasm lines of St. John’s wort (SJW; Hypericum perforatum L.) selected for enhanced hypericin and hyperforin content were evaluated for potential activity against colon cancer. Bioactivity was assessed in signaling pathways of tumor necrosis factor-a (TNF-?) and nuclear transcription factor-?B (NF-?B) in HT-29 colon cancer cells. Both extracts and the hypericin standard significantly inhibited growth of HT-29 cells. Levels of active NF-?B were reduced in cells treated with either of the plant extracts or hypericin, but the purified hyperforin standard was comparatively ineffective. The combination of TNF-? and SJW treatments had significantly higher cytotoxic effects, and reduced the expression of NF-?B, inhibitor of NF-?Bs (I?Ba), I?B kinase b (IKKb), and TNF receptor-1. These observations indicate the potential of SJW as a source of cancer therapies, including those that act synergistically with TNF-?. The phytochemical complexity of SJW tissues necessitates consistent, optimized plant extracts for optimal results and the data indicate that additional, possibly unidentified, phytochemicals from SJW have potential in the treatment or prevention of colon cancer.

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

Full frame distilled prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. Learned from the 10,348 direct Codex labels and 10,348 direct Gemma labels. Candidate is the union of thresholded teacher heads; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels or direct frontier model labels.

metaresearch head score (Codex)0.000
metaresearch head score (Gemma)0.000
Version: codex-gemma-dda1882f352aValidation status: machine_predicted_unvalidated
Candidate categoriesnone
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Bench or experimental · Consensus signal: Bench or experimental
GenreCandidate signal: Empirical · Consensus signal: Empirical
Teacher disagreement score0.104
Threshold uncertainty score0.474

Codex and Gemma teacher scores by category

CategoryCodexGemma
Metaresearch0.0000.000
Meta-epidemiology (narrow)0.0000.000
Meta-epidemiology (broad)0.0010.000
Bibliometrics0.0000.000
Science and technology studies0.0000.000
Scholarly communication0.0000.000
Open science0.0000.000
Research integrity0.0000.000
Insufficient payload (model declined to judge)0.0000.000

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.013
GPT teacher head0.287
Teacher spread0.274 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it