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Record W2084532091 · doi:10.1139/v01-037

Synthesis and coordination studies of new aminoalcohol functionalized tertiary phosphines

2001· article· en· W2084532091 on OpenAlexvenueno aff
S.E. Durran, Martin B. Smith, Alexandra M. Z. Slawin, Thomas Gelbrich, Michael B. Hursthouse, Mark E. Light

Bibliographic record

VenueCanadian Journal of Chemistry · 2001
Typearticle
Languageen
FieldMedicine
TopicMetal complexes synthesis and properties
Canadian institutionsnot available
Fundersnot available
KeywordsChemistryPhosphineLigand (biochemistry)Medicinal chemistryStereochemistryMetalAqueous solutionTransition metalNuclear magnetic resonance spectroscopyCatalysisOrganic chemistry

Abstract

fetched live from OpenAlex

The synthesis of two new aminoalcohol functionalized tertiary phosphines o-Ph 2 PCH 2 N(H)C 6 H 4 (OH) (I) and o-Ph 2 PCH 2 N(H)C 6 H 4 (CH 2 OH) (II) are reported. Oxidation with aqueous H 2 O 2 gave the corresponding phosphine oxides o-Ph 2 P(O)CH 2 N(H)C 6 H 4 (OH) (III) and o-Ph 2 P(O)CH 2 N(H)C 6 H 4 (CH 2 OH) (IV) ( 31 P NMR evidence only). The ligating ability of I, II and, in several cases, the known ligand 2,3-Ph 2 PCH 2 N(H)C 5 H 3 N(OH) (V), was investigated with a range of late transition-metal precursors. Accordingly, reaction of 2 equiv of I (or II) with [MCl 2 (cod)] (M = Pd or Pt, cod = cycloocta-1,5-diene) gave the corresponding dichloro metal(II) complexes [MCl 2 (I) 2 ] (M = Pd 1; M = Pt 2) and [MCl 2 (II) 2 ] (M = Pd 3; M = Pt 4) in which I (and II) P-coordinate. Solution NMR studies reveal that 2 and 4 are exclusively cis whereas 1 and 3 are present as a mixture of cis and (or) trans isomers [4.7:1 (for 1); 2.2:1 (for 3)]. Reaction of 2 equiv of II with [Pt(CH 3 ) 2 (cod)] gave the neutral complex [Pt(CH 3 ) 2 (II) 2 ] (5) whose X-ray structure confirmed a cis disposition of "hybrid" ligands. In contrast, reaction of I with [Pt(CH 3 ) 2 (cod)] gave initially [Pt(CH 3 ) 2 (I) 2 ] (6) which, upon standing, afforded several products possibly reflecting an increased acidity of the phenolic groups of ligated I. Chloro bridge cleavage reactions of [{Ru(µ-Cl)Cl(p-cymene)} 2 ] or [{Rh(µ-Cl)Cl{C 5 (CH 3 ) 5 }} 2 ] with I (or II) proceeds smoothly and gave the mononuclear complexes [RuCl 2 (p-cymene)I] (7), [RuCl 2 (p-cymene)II] (8), [RhCl 2 {C 5 (CH 3 ) 5 }I] (9), and [RhCl 2 {C 5 (CH 3 ) 5 }II] (10) in good yield. X-ray crystallography confirms both ruthenium complexes bear P-coordinated I (or II) ligands. Molecules of 7 are linked into linear chains via O-H···Cl coord intermolecular hydrogen bonding, a feature absent in the closely related compound 8. Reaction of [AuCl(tht)] (tht = tetrahydrothiophene) with 1 equiv of I (or II) gave the corresponding gold(I) complexes [AuCl(I)] (11) and [AuCl(II)] (12). Bridge cleavage of the cyclometallated palladium(II) dimers [{Pd(µ-Cl)(C~N)} 2 ] [C~N = C,N-C 6 H 4 CH 2 N(CH 3 ) 2 , C,N-C 10 H 6 N(CH 3 ) 2 , C,N-C 6 H 4 N=NC 6 H 5 ] with V (or I) gave the neutral complexes [PdCl(C~N)V] (13-15) (or [PdCl(C 9 H 12 N)I] (16)), respectively. Chloride abstraction from 13 (or 15) with Ag[BF 4 ] gave the cationic complexes [Pd(C~N)V][BF 4 ] (17) (or 18) in which V P,N pyridyl -chelates to the palladium(II) metal centre. The X-ray structures of 13 and 18 have been determined and confirm the expected coordination environments. An array of intra- and intermolecular H-bonding contacts are also observed. All compounds have been characterized by a combination of spectroscopic and analytical studies.Key words: phosphines, crystal structures, alcohols, precious metals.

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

How this classification was reachedexpand

Full frame distilled prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. Learned from the 10,348 direct Codex labels and 10,348 direct Gemma labels. Candidate is the union of thresholded teacher heads; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels or direct frontier model labels.

metaresearch head score (Codex)0.000
metaresearch head score (Gemma)0.001
Version: codex-gemma-dda1882f352aValidation status: machine_predicted_unvalidated
Candidate categoriesnone
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Bench or experimental · Consensus signal: Bench or experimental
GenreCandidate signal: Empirical · Consensus signal: Empirical
Teacher disagreement score0.096
Threshold uncertainty score0.909

Codex and Gemma teacher scores by category

CategoryCodexGemma
Metaresearch0.0000.001
Meta-epidemiology (narrow)0.0000.000
Meta-epidemiology (broad)0.0000.000
Bibliometrics0.0000.000
Science and technology studies0.0000.000
Scholarly communication0.0000.000
Open science0.0000.000
Research integrity0.0000.000
Insufficient payload (model declined to judge)0.0010.000

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.059
GPT teacher head0.272
Teacher spread0.214 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it

Classification

machine, unvalidated

Machine predicted; a candidate call from one teacher head, not a consensus.

The models applied no category: nothing in the taxonomy fit this work.
Study designBench or experimental
Domainnot available
GenreEmpirical

How this classification was reached, model by model and score by score, is at the end of the page under "How this classification was reached".

Quick stats

Citations26
Published2001
Admission routes1
Has abstractyes

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