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Record W2084802551 · doi:10.1021/jp002622c

Complexation Dynamics of Xanthone and Thioxanthone to β-Cyclodextrin Derivatives

2001· article· en· W2084802551 on OpenAlexaff
Laura T. Okano, T. C. Barros, Doug T. H. Chou, Andrew J. Bennet, Cornelia Bohne

Bibliographic record

VenueThe Journal of Physical Chemistry B · 2001
Typearticle
Languageen
FieldPharmacology, Toxicology and Pharmaceutics
TopicDrug Solubulity and Delivery Systems
Canadian institutionsUniversity of VictoriaSimon Fraser University
Fundersnot available
KeywordsThioxanthoneXanthoneChemistryMoietyExcited statePhotochemistryBinding constantReaction rate constantEquilibrium constantTriplet stateDissociation constantStereochemistryCrystallographyKineticsBinding sitePhysical chemistryMoleculeOrganic chemistryPhotoinitiatorMonomer

Abstract

fetched live from OpenAlex

The complexation dynamics of xanthone to substituted β-cyclodextrins (CDs) and of thioxanthone to β-CD was studied by directly following the relocation of the excited triplet-state ketones from the CD cavity to the aqueous phase. Equilibrium constants for the ground-state complexation of both ketones with CDs were determined from fluorescence studies. The complexation efficiency and dynamics of thioxanthone with β-CD were the same as previously observed for the xanthone/β-CD system. Substitution of some of the hydrogens on the alcohol groups by methyl moieties at both entrances to the β-CD cavity increased the equilibrium constant for ground-state xanthone, but decreased that for the excited triplet state, leading to a larger difference for the binding behavior of these two electronic states of the guest. Addition of one pendant arm containing a carboxyl moiety to the rim where xanthone is bound does not change the binding efficiency of the ground state or the binding dynamics of triplet xanthone. In contrast, when this arm contains an ethyl ester moiety, the binding efficiencies of both the ground and excited triplet states are increased. The higher binding constant for triplet xanthone is due to an increase of the association rate constant and a decrease for the dissociation rate constant.

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

How this classification was reachedexpand

Full frame distilled prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. Learned from the 10,348 direct Codex labels and 10,348 direct Gemma labels. Candidate is the union of thresholded teacher heads; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels or direct frontier model labels.

metaresearch head score (Codex)0.001
metaresearch head score (Gemma)0.000
Version: codex-gemma-dda1882f352aValidation status: machine_predicted_unvalidated
Candidate categoriesnone
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Bench or experimental · Consensus signal: Bench or experimental
GenreCandidate signal: Empirical · Consensus signal: Empirical
Teacher disagreement score0.094
Threshold uncertainty score0.324

Codex and Gemma teacher scores by category

CategoryCodexGemma
Metaresearch0.0010.000
Meta-epidemiology (narrow)0.0000.000
Meta-epidemiology (broad)0.0000.000
Bibliometrics0.0000.000
Science and technology studies0.0000.000
Scholarly communication0.0000.000
Open science0.0000.000
Research integrity0.0000.000
Insufficient payload (model declined to judge)0.0000.000

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.071
GPT teacher head0.396
Teacher spread0.325 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it

Classification

machine, unvalidated

Machine predicted; a candidate call from one teacher head, not a consensus.

The models applied no category: nothing in the taxonomy fit this work.
Study designBench or experimental
Domainnot available
GenreEmpirical

How this classification was reached, model by model and score by score, is at the end of the page under "How this classification was reached".

Quick stats

Citations44
Published2001
Admission routes1
Has abstractyes

Explore more

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