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Record W2318502144 · doi:10.1021/om201288p

Reactions of Grubbs Catalysts with Excess Methoxide: Formation of Novel Methoxyhydride Complexes

2012· article· en· W2318502144 on OpenAlex

Why this work is in the frame

A frame that forgets how it found something cannot be audited. These are the routes that admitted this work.

affAt least one author lists a Canadian institution in the pinned OpenAlex snapshot.

Bibliographic record

VenueOrganometallics · 2012
Typearticle
Languageen
FieldChemistry
TopicSynthetic Organic Chemistry Methods
Canadian institutionsUniversity of Ottawa
Fundersnot available
KeywordsChemistryMetathesisMethoxideMedicinal chemistryIMesAdductDecarbonylationLigand (biochemistry)PhosphineCatalysisSodium methoxideRutheniumStereochemistryCarbeneOrganic chemistryReceptorPolymerization

Abstract

fetched live from OpenAlex

On exposure to NaOMe (≥3 equiv) in CH 2 Cl 2 –MeOH at 23 °C, the first-generation Grubbs catalyst RuCl 2 (PCy 3 ) 2 (═CHPh) ( 1a ) is immediately transformed into the six-coordinate methoxyhydride complexes RuH(OMe)(CO) 2 (PCy 3 ) 2 ( 4a ) and RuH(OMe)(CO)(H 2 )(PCy 3 ) 2 ( 5a ). Complex 5a can be recycled into 4a under conditions conducive to removal of H 2 . The second-generation catalyst RuCl 2 (IMes)(PCy 3 )(═CHPh) ( 1b; IMes = N,N ′-bis(mesityl)imidazol-2-ylidene) reacts more slowly, requiring several hours even at 20 equiv of NaOMe, and terminates at five-coordinate RuH(OMe)(CO)(IMes)(PCy 3 ) ( 3b ). Experiments in the presence of added PCy 3 reveal that consumption of 1a, but not 1b, proceeds via the four-coordinate intermediate formed by equilibrium loss of phosphine, a function of the lability of the PCy 3 ligand at ambient temperatures. The poor accessibility of such an intermediate for 1b at 23 °C retards salt metathesis and inhibits further reaction of 3b . For the bis(PCy 3 ) analogue 3a, fast transformation into 4a is proposed to involve reversible loss of PCy 3, coordination of methanol, σ-metathesis of methanol at the hydride site to liberate H 2, and β-elimination/decarbonylation of bound methoxide. Competitive uptake of H 2 by 3a yields six-coordinate 5a (the dihydrogen adduct of 3a ). Independent routes to RuH(OMe)(CO) 2 (L)(PCy 3 ) ( 4a/b; a, L = PCy 3; b, L = IMes) were developed: these involved sequential transformation of RuHCl(CO)(L)(PCy 3 ) ( 2a/b ) into the bis-carbonyl adducts RuHCl(CO) 2 (L)(PCy 3 ) ( 7a/b ) under CO, conversion of 7a/b into the more reactive triflates RuH(OTf)(CO) 2 (L)(PCy 3 ) ( 8a/b ), and reaction of 8a/b with equimolar NaOMe. Dihydride 6b was also prepared, by reaction of 8b with NaH.

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

Full frame distilled prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. Learned from the 10,348 direct Codex labels and 10,348 direct Gemma labels. Candidate is the union of thresholded teacher heads; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels or direct frontier model labels.

metaresearch head score (Codex)0.001
metaresearch head score (Gemma)0.001
Version: codex-gemma-dda1882f352aValidation status: machine_predicted_unvalidated
Candidate categoriesInsufficient payload (model declined to judge)
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Bench or experimental · Consensus signal: Bench or experimental
GenreCandidate signal: Empirical · Consensus signal: Empirical
Teacher disagreement score0.022
Threshold uncertainty score1.000

Codex and Gemma teacher scores by category

CategoryCodexGemma
Metaresearch0.0010.001
Meta-epidemiology (narrow)0.0000.000
Meta-epidemiology (broad)0.0010.000
Bibliometrics0.0000.001
Science and technology studies0.0000.000
Scholarly communication0.0000.000
Open science0.0000.000
Research integrity0.0000.000
Insufficient payload (model declined to judge)0.0010.000

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.050
GPT teacher head0.303
Teacher spread0.253 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it