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Record W2488539909 · doi:10.1385/0-89603-078-4:139

Muscarinic Cholinergic Receptors

2003· book-chapter· en· W2488539909 on OpenAlexaff
Andrew P. Braun, Prakash V. Sulakhe

Bibliographic record

VenueHumana Press eBooks · 2003
Typebook-chapter
Languageen
FieldBiochemistry, Genetics and Molecular Biology
TopicReceptor Mechanisms and Signaling
Canadian institutionsUniversity of Saskatchewan
Fundersnot available
KeywordsMuscarinic acetylcholine receptorCholinergicNicotinic agonistNeuroscienceAcetylcholineAcetylcholine receptorNeurotransmitter receptorMuscarinic acetylcholine receptor M4Muscarinic acetylcholine receptor M5BiologyReceptorNeurotransmitterPopulationMuscarinic acetylcholine receptor M2Cholinergic neuronCentral nervous systemEndocrinologyMuscarinic acetylcholine receptor M3Internal medicineMedicineBiochemistry

Abstract

fetched live from OpenAlex

In the central nervous system (CNS), modulation of neuronal activity is brought about by the actions of endogenous “neurotransmitters” that specifically interact with receptor proteins located in the neuronal cell membrane. In the cholinergic system, acetylcholine is the primary neurotransmitter released in the CNS, and appears to alter neuronal excitability by affecting such processes as cGMP production and K+ flux (Heilbronn and Bartfai, 1978). In contrast to the periphery, in which the cholinergic receptor population is divided between nicotinic and muscarinic subclasses, the CNS-associated cholinergic receptor appears to be predominantly of the muscarinic type, although there is evidence that the spinal cord contains substantial amounts of nicotinic receptors (Heilbronn and Bartfai, 1978). Historically, the initial characterization of cholinergic actions was provided by A. S. V. Burgen. Although these early studies, using smooth muscle tissue (Burgen and Spero, 1968; Burgen et al., 1974), provided initial clues about the peripheral muscarinic receptors, since then there have been numerous investigations, especially following the advent of radioligand binding assays, from which have come many novel observations of physiological significance.

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

How this classification was reachedexpand

Full frame distilled prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. Learned from the 10,348 direct Codex labels and 10,348 direct Gemma labels. Candidate is the union of thresholded teacher heads; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels or direct frontier model labels.

metaresearch head score (Codex)0.000
metaresearch head score (Gemma)0.000
Version: codex-gemma-dda1882f352aValidation status: machine_predicted_unvalidated
Candidate categoriesMeta-epidemiology (narrow)
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Not applicable · Consensus signal: none
GenreCandidate signal: Other · Consensus signal: Other
Teacher disagreement score0.777
Threshold uncertainty score1.000

Codex and Gemma teacher scores by category

CategoryCodexGemma
Metaresearch0.0000.000
Meta-epidemiology (narrow)0.0000.001
Meta-epidemiology (broad)0.0000.000
Bibliometrics0.0000.000
Science and technology studies0.0000.000
Scholarly communication0.0000.000
Open science0.0000.000
Research integrity0.0010.000
Insufficient payload (model declined to judge)0.0010.000

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.039
GPT teacher head0.247
Teacher spread0.208 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it

Classification

machine, unvalidated

Machine predicted; a candidate call from one teacher head, not a consensus.

Study designNot applicable
Domainnot available
GenreOther

How this classification was reached, model by model and score by score, is at the end of the page under "How this classification was reached".

Quick stats

Citations21
Published2003
Admission routes1
Has abstractyes

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