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Record W2514299705 · doi:10.1021/acs.cgd.6b01088

Reevaluating the Stability and Prevalence of Conglomerates: Implications for Preferential Crystallization

2016· article· en· W2514299705 on OpenAlex
Alberto Otero‐de‐la‐Roza, Jason E. Hein, Erin R. Johnson

Why this work is in the frame

A frame that forgets how it found something cannot be audited. These are the routes that admitted this work.

affAt least one author lists a Canadian institution in the pinned OpenAlex snapshot.
fundA Canadian funder is recorded on the work.

Bibliographic record

VenueCrystal Growth & Design · 2016
Typearticle
Languageen
FieldMaterials Science
TopicCrystallization and Solubility Studies
Canadian institutionsDalhousie UniversityOkanagan University CollegeUniversity of British Columbia, Okanagan CampusUniversity of British Columbia
FundersDivision of ChemistryNational Science FoundationNational Cancer InstituteNatural Sciences and Engineering Research Council of CanadaMinisterio de Ciencia e InnovaciónWestern Canada Research Grid
KeywordsCrystallizationChemistryEnantiomerPhase (matter)CrystallographyChiral resolutionCrystal (programming language)ThermodynamicsDispersion (optics)StereochemistryPhysicsOrganic chemistryQuantum mechanics

Abstract

fetched live from OpenAlex

Chiral resolution by preferential crystallization from a racemic or scalemic solution occurs by selective crystallization of a single enantiomer as a homochiral solid phase, known as a conglomerate. However, there is a prevailing perception that stable homochiral crystals are quite rare and are estimated to form in only 5–10% of all chiral compounds. In this work, the prevalence rate of stable conglomerates is reexamined using dispersion-corrected density-functional theory calculations for a collection of homochiral and heterochiral crystal pairs. The homochiral crystal is found to be the thermodynamically stable phase for 19% of the examined compounds. This value represents a lower bound of the prevalence rate since our sample is necessarily biased because the comparison is limited to cases where a stable heterochiral phase exists and does not include molecules with no reported heterochiral phase. Even so, this lower bound is two to four times higher than the often-quoted conglomerate prevalence rate, a value that is also based on (experimental) thermodynamic quantities. In addition, our results are used to reexamine Wallach’s rule and the close-packing principle. It is concluded that the prevalence of stable conglomerates has been underestimated, and, provided thermodynamic equilibrium drives the crystallization process, preferential crystallization has a much wider scope of applicability than previously assumed.

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

Full frame distilled prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. Learned from the 10,348 direct Codex labels and 10,348 direct Gemma labels. Candidate is the union of thresholded teacher heads; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels or direct frontier model labels.

metaresearch head score (Codex)0.001
metaresearch head score (Gemma)0.002
Version: codex-gemma-dda1882f352aValidation status: machine_predicted_unvalidated
Candidate categoriesnone
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Bench or experimental · Consensus signal: Bench or experimental
GenreCandidate signal: Empirical · Consensus signal: none
Teacher disagreement score0.671
Threshold uncertainty score0.334

Codex and Gemma teacher scores by category

CategoryCodexGemma
Metaresearch0.0010.002
Meta-epidemiology (narrow)0.0000.000
Meta-epidemiology (broad)0.0000.000
Bibliometrics0.0000.000
Science and technology studies0.0000.000
Scholarly communication0.0000.000
Open science0.0000.000
Research integrity0.0000.000
Insufficient payload (model declined to judge)0.0000.000

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.090
GPT teacher head0.301
Teacher spread0.211 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it