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Record W2560312435 · doi:10.1016/j.celrep.2016.11.014

Multivalent Histone and DNA Engagement by a PHD/BRD/PWWP Triple Reader Cassette Recruits ZMYND8 to K14ac-Rich Chromatin

2016· article· en· W2560312435 on OpenAlexafffund
P. Savitsky, T. Krojer, Takao Fujisawa, Jean‐Philippe Lambert, S. Picaud, Chen Yi Wang, Erin K. Shanle, Krzysztof Krajewski, Hans Friedrichsen, Alexander Kanapin, Colin R. Goding, Matthieu Schapira, Anastasia Samsonova, Brian D. Strahl, Anne‐Claude Gingras, P. Filippakopoulos

Bibliographic record

VenueCell Reports · 2016
Typearticle
Languageen
FieldBiochemistry, Genetics and Molecular Biology
TopicProtein Degradation and Inhibitors
Canadian institutionsUniversity of TorontoStructural Genomics ConsortiumLunenfeld-Tanenbaum Research InstituteMount Sinai Hospital
FundersEshelman Institute for Innovation, University of North Carolina at Chapel HillJanssen PharmaceuticalsOntario Genomics InstituteNational Institute of General Medical SciencesMedical Research Council CanadaMedical Research CouncilTakeda CanadaNational Institutes of HealthOntario Ministry of Economic Development and InnovationMerckWellcomeGovernment of CanadaShenzhen Gas CorporationUehara Memorial FoundationWellcome TrustCanada Foundation for InnovationLudwig Institute for Cancer ResearchGenome CanadaAbbVieNovartis PharmaBoehringer IngelheimCanadian Institutes of Health ResearchInnovative Medicines InitiativePfizer
KeywordsChromatinHistoneDNANucleosomeCell biologyChemistryFlexibility (engineering)Computational biologyGeneticsBiology

Abstract

fetched live from OpenAlex

Elucidation of interactions involving DNA and histone post-translational-modifications (PTMs) is essential for providing insights into complex biological functions. Reader assemblies connected by flexible linkages facilitate avidity and increase affinity; however, little is known about the contribution to the recognition process of multiple PTMs because of rigidity in the absence of conformational flexibility. Here, we resolve the crystal structure of the triple reader module (PHD-BRD-PWWP) of ZMYND8, which forms a stable unit capable of simultaneously recognizing multiple histone PTMs while presenting a charged platform for association with DNA. Single domain disruptions destroy the functional network of interactions initiated by ZMYND8, impairing recruitment to sites of DNA damage. Our data establish a proof of principle that rigidity can be compensated by concomitant DNA and histone PTM interactions, maintaining multivalent engagement of transient chromatin states. Thus, our findings demonstrate an important role for rigid multivalent reader modules in nucleosome binding and chromatin function.

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

How this classification was reachedexpand

Full frame distilled prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. Learned from the 10,348 direct Codex labels and 10,348 direct Gemma labels. Candidate is the union of thresholded teacher heads; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels or direct frontier model labels.

metaresearch head score (Codex)0.000
metaresearch head score (Gemma)0.000
Version: codex-gemma-dda1882f352aValidation status: machine_predicted_unvalidated
Candidate categoriesnone
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Bench or experimental · Consensus signal: Bench or experimental
GenreCandidate signal: Empirical · Consensus signal: Empirical
Teacher disagreement score0.202
Threshold uncertainty score0.608

Codex and Gemma teacher scores by category

CategoryCodexGemma
Metaresearch0.0000.000
Meta-epidemiology (narrow)0.0000.000
Meta-epidemiology (broad)0.0000.000
Bibliometrics0.0000.000
Science and technology studies0.0000.000
Scholarly communication0.0000.000
Open science0.0000.000
Research integrity0.0000.000
Insufficient payload (model declined to judge)0.0000.000

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.020
GPT teacher head0.267
Teacher spread0.246 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it

Classification

machine, unvalidated

Machine predicted; a candidate call from one teacher head, not a consensus.

The models applied no category: nothing in the taxonomy fit this work.
Study designBench or experimental
Domainnot available
GenreEmpirical

How this classification was reached, model by model and score by score, is at the end of the page under "How this classification was reached".

Quick stats

Citations104
Published2016
Admission routes2
Has abstractyes

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