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Record W2595647287 · doi:10.1021/jacs.6b12607

Generation of Hydrofluoronickelacycles from Trifluoroethylene and Ni(0): Ligand Effects on Regio-/Stereoselectivity and Reactivity

2017· article· en· W2595647287 on OpenAlexafffund
Kaitie A. Giffin, Lorraine A. Pua, Sarah Piotrkowski, Bulat Gabidullin, Ilia Korobkov, Russell P. Hughes, R. Tom Baker

Bibliographic record

VenueJournal of the American Chemical Society · 2017
Typearticle
Languageen
FieldPharmacology, Toxicology and Pharmaceutics
TopicFluorine in Organic Chemistry
Canadian institutionsUniversity of Ottawa
FundersNatural Sciences and Engineering Research Council of CanadaCanada Research ChairsOntario Ministry of Economic Development and InnovationUniversity of Ottawa
KeywordsChemistryStereoselectivityYield (engineering)Reactivity (psychology)Ligand (biochemistry)BromideCis–trans isomerismMedicinal chemistryStereochemistryLewis acids and basesCatalysisOrganic chemistry

Abstract

fetched live from OpenAlex

Treatment of Ni(0) complexes 1a – e with sub-atmospheric pressures of trifluoroethylene (TrFE) affords hydrofluoronickelacyclopentanes L 2 Ni(C 4 F 6 H 2 ) 2a – e (L = PPh 3, P(O- o -tol) 3, PPh 2 Me, PPhMe 2, PMe 3 ). Fluorine NMR analysis of 2a – e demonstrates predominant formation of three (of the possible six) isomers upon oxidative cycloaddition of TrFE: the cis and trans head–tail isomers and the trans head–head isomer, where the CHF group is defined as the TrFE “head”. The respective ratios of L 2 Ni(C 4 F 6 H 2 ) isomers are influenced by the nature of L, with smaller phosphines favoring the thermodynamically preferred (from DFT calculations) trans head–head isomer (cf. 50% with PMe 3 ) and the largest affording small amounts of the tail–tail isomers. Lewis and Brønsted acids induce a surprising double C–F bond activation in 2c – d, affording small functionalized hydrofluoroalkenes. Interestingly, varying the acid employed dictates the organic product obtained from the head–tail isomers: BF 3 ·OEt 2 is selective for 1,1,2,3-tetrafluorocyclobutene, whereas Me 3 SiOTf and N,N -dimethylanilinium bromide yield ( Z,E )-1,1,3,4-tetrafluorobutadiene as the major fluorinated product. Reaction intermediates were isolated, and possible pathways are discussed.

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

How this classification was reachedexpand

Full frame machine prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. The Gemma side is a direct model label for every work in the frame, read from the title-only record. The Codex side is a classifier learned from the 10,348 direct Codex labels and calibrated to design-weighted sample rates; fields without enough sample support carry no Codex call. Candidate is the union of the two sides; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels.

metaresearch head score (Codex)0.000
metaresearch head score (Gemma)0.000
Version: metacan-v3-hybrid-931329e0061cValidation status: machine_predicted_unvalidated
Candidate categoriesnone
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Bench or experimental · Consensus signal: Bench or experimental
GenreCandidate signal: Empirical · Consensus signal: Empirical
Teacher disagreement score0.003
Threshold uncertainty score0.010

Distilled classifier scores by category (both heads)

CategoryCodexGemma
Metaresearch0.0000.000
Meta-epidemiology (narrow)0.0000.000
Meta-epidemiology (broad)0.0000.000
Bibliometrics0.0000.000
Science and technology studies0.0000.000
Scholarly communication0.0000.000
Open science0.0000.000
Research integrity0.0000.000
Insufficient payload (model declined to judge)0.0030.001

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.065
GPT teacher head0.380
Teacher spread0.316 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it

Classification

machine, unvalidated

Machine predicted; a candidate call from one source (direct Gemma or distilled Codex), not a consensus.

The models applied no category: nothing in the taxonomy fit this work.
Study designBench or experimental
Domainnot available
GenreEmpirical

How this classification was reached, model by model and score by score, is at the end of the page under "How this classification was reached".

Quick stats

Citations19
Published2017
Admission routes2
Has abstractyes

Explore more

Same venueJournal of the American Chemical SocietySame topicFluorine in Organic ChemistryFrench-language works237,207