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Record W2845742321 · doi:10.1021/acs.organomet.8b00297

β-Hydrogen Elimination and Reductive Elimination from a κ<sup>3</sup>-PPC Nickel Complex

2018· article· en· W2845742321 on OpenAlexafffund
Amanda C. Zimmerman, Michael D. Fryzuk

Bibliographic record

VenueOrganometallics · 2018
Typearticle
Languageen
FieldChemistry
TopicAsymmetric Hydrogenation and Catalysis
Canadian institutionsUniversity of British Columbia
FundersNatural Sciences and Engineering Research Council of Canada
KeywordsChemistryReductive eliminationOxidative additionMedicinal chemistryElimination reactionNickelArylLigand (biochemistry)ReagentHeteroatomInorganic chemistryOrganic chemistryCatalysisRing (chemistry)

Abstract

fetched live from OpenAlex

The incorporation of a PPC donor ligand set onto nickel is described. While C–H activation routes using Ni(II) precursors and benzyl- and phenethyl-substituted diphosphines But2PCH2CH2P(But)R failed, success was achieved via oxidative addition of the 2-bromo-benzyl-ligand precursor But2PCH2CH2P(But)(CH2-o-C6H4Br) with Ni(COD)2 to generate [κ3-BnPPC]NiBr. Subsequent reaction with KBEt3H resulted in decomposition unless PPh3 was present, which allowed isolation of the tricoordinate Ni(0) complex [κ2-BnPP]Ni(PPh3). Reaction of [κ3-BnPPC]NiBr with EtMgCl also resulted in the formation of the Ni(0) ethylene complex, [κ2-BnPP]Ni(η2-C2H4), via β-elimination followed by reductive elimination. Deuterium-labeling studies are consistent with a reversible β-elimination process prior to reductive elimination, which scrambles the deuterium isotopes. Reaction of [κ3-BnPPC]NiBr with CH3Li results in the formation of the Ni(II) methyl complex, [κ3-BnPPC]Ni(CH3). Heating this species in the presence of PPh3 results in the formation of the Ni(0) derivative, [κ2-Bn-o-MePP]Ni(PPh3), in which reductive elimination of the methyl and aryl units has occurred. Reaction of [κ3-BnPPC]NiBr with heteroatom-containing species such as sodium isopropoxide, sodium 2-propanethiolate, and lithium methylphenylamide resulted in different outcomes depending on the heteroatom; with isopropoxide, the products isolated were geometric isomers of Ni(0) η2-acetone adducts, which presumably arise via a β-elimination–reductive elimination sequence; the analogous sulfur reagent generated isolable Ni(II) isopropyl thiolate species that was resistant to β-elimination upon thermolysis; with methylphenylamide, the Ni(II) amido complex could be isolated and structurally characterized; subsequent heating to 80 °C resulted in β-elimination followed by reductive elimination to generate a Ni(0) phenylimine complex. While the κ3-PPC donor set generates stable Ni(II) derivatives, further functionalization at nickel with hydride, alkyl, and heteroatom-containing moieties can lead to Ni(0) products via a combination of β-elimination and/or reductive elimination.

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

How this classification was reachedexpand

Full frame distilled prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. Learned from the 10,348 direct Codex labels and 10,348 direct Gemma labels. Candidate is the union of thresholded teacher heads; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels or direct frontier model labels.

metaresearch head score (Codex)0.000
metaresearch head score (Gemma)0.000
Version: codex-gemma-dda1882f352aValidation status: machine_predicted_unvalidated
Candidate categoriesMeta-epidemiology (narrow), Insufficient payload (model declined to judge)
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Bench or experimental · Consensus signal: Bench or experimental
GenreCandidate signal: Empirical · Consensus signal: Empirical
Teacher disagreement score0.329
Threshold uncertainty score1.000

Codex and Gemma teacher scores by category

CategoryCodexGemma
Metaresearch0.0000.000
Meta-epidemiology (narrow)0.0000.000
Meta-epidemiology (broad)0.0000.000
Bibliometrics0.0000.001
Science and technology studies0.0000.000
Scholarly communication0.0000.000
Open science0.0000.000
Research integrity0.0000.000
Insufficient payload (model declined to judge)0.0060.000

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.019
GPT teacher head0.245
Teacher spread0.226 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it

Classification

machine, unvalidated

Machine predicted; a candidate call from one teacher head, not a consensus.

Study designBench or experimental
Domainnot available
GenreEmpirical

How this classification was reached, model by model and score by score, is at the end of the page under "How this classification was reached".

Quick stats

Citations10
Published2018
Admission routes2
Has abstractyes

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