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Record W3200833013 · doi:10.26434/chemrxiv.9914378.v1

A Diversified Machine Learning Strategy for Predicting and Understanding Molecular Melting Points

2019· preprint· en· W3200833013 on OpenAlexaff
Ganesh Sivaraman, Nicholas E. Jackson, Benjamín Sánchez-Lengeling, Álvaro Vázquez‐Mayagoitia, Alán Aspuru‐Guzik, Venkatram Vishwanath, Juan Pablo

Bibliographic record

VenueChemRxiv · 2019
Typepreprint
Languageen
FieldComputer Science
TopicComputational Drug Discovery Methods
Canadian institutionsVector InstituteUniversity of TorontoCanadian Institute for Advanced Research
FundersArgonne National LaboratoryOffice of ScienceU.S. Department of Energy
KeywordsAutoencoderComputer scienceMolecular graphCluster analysisEmbeddingGraphMachine learningArtificial intelligenceArtificial neural networkUnsupervised learningQuantum chemicalGaussianData miningTheoretical computer scienceMoleculeChemistryComputational chemistry

Abstract

fetched live from OpenAlex

The ability to predict multi-molecule processes, using only knowledge of single molecule structure, stands as a grand challenge for molecular modeling. Methods capable of predicting melting points (MP) solely from chemical structure represent a canonical example, and are highly desirable in many crucial industrial applications. In this work, we explore a data-driven approach utilizing machine learning (ML) techniques to predict and understand the MP of molecules. Several experimental databases are aggregated from the literature to design a low-bias dataset that includes 3D structural and quantum-chemical properties. Using experimental and polymorph-induced uncertainties, we derive a tenable lower limit for MP prediction accuracy, and apply graph neural networks and Gaussian processes to predict MP competitive with these error bounds. To further understand how MP correlates with molecular structure, we employ several semi-supervised and unsupervised ML techniques. First, we use unsupervised clustering methods to identify classes of molecules, their common fragments, and expected errors for each data set. We then build molecular geometric spaces shaped by MP with a semi-supervised variational autoencoder and graph embedding spaces, and apply graph attribution methods to highlight atom-level contributions to MP within the datasets. Overall, this work serves as a case study of how to employ a diversified ML toolkit to predict and understand correlations between molecular structures and thermophysical properties of interest.

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

How this classification was reachedexpand

Full frame distilled prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. Learned from the 10,348 direct Codex labels and 10,348 direct Gemma labels. Candidate is the union of thresholded teacher heads; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels or direct frontier model labels.

metaresearch head score (Codex)0.001
metaresearch head score (Gemma)0.000
Version: codex-gemma-dda1882f352aValidation status: machine_predicted_unvalidated
Candidate categoriesMeta-epidemiology (narrow)
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Simulation or modeling · Consensus signal: Simulation or modeling
GenreCandidate signal: Empirical · Consensus signal: none
Teacher disagreement score0.778
Threshold uncertainty score1.000

Codex and Gemma teacher scores by category

CategoryCodexGemma
Metaresearch0.0010.000
Meta-epidemiology (narrow)0.0000.000
Meta-epidemiology (broad)0.0000.000
Bibliometrics0.0000.000
Science and technology studies0.0000.000
Scholarly communication0.0000.000
Open science0.0010.002
Research integrity0.0000.001
Insufficient payload (model declined to judge)0.0000.000

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.090
GPT teacher head0.319
Teacher spread0.229 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it

Classification

machine, unvalidated

Machine predicted; a candidate call from one teacher head, not a consensus.

Study designSimulation or modeling
Domainnot available
GenreEmpirical

How this classification was reached, model by model and score by score, is at the end of the page under "How this classification was reached".

Quick stats

Citations4
Published2019
Admission routes1
Has abstractyes

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