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Record W4296896604 · doi:10.3389/fphar.2022.1019004

Editorial: Emerging perspectives in sodium channelopathies

2022· editorial· en· W4296896604 on OpenAlexaff
James R. Groome, H. J. Ray, Mohamed Chahine

Bibliographic record

VenueFrontiers in Pharmacology · 2022
Typeeditorial
Languageen
FieldBiochemistry, Genetics and Molecular Biology
TopicIon channel regulation and function
Canadian institutionsUniversité Laval
FundersNational Institute of General Medical Sciences
KeywordsSodium channelClinical pharmacologyPharmacologyMedicineIon channelNeuroscienceChemistrySodiumPsychologyInternal medicineReceptor

Abstract

fetched live from OpenAlex

Emerging perspectives in sodium channelopathiesRecent advances in molecular biology have greatly increased our understanding of ion channel structure and function.Cloning of genes encoding voltage-gated ion channels expanded the investigation of action potential signaling in neurons and muscle fibers.Gene sequences predicted the crucial role of positively charged residues in S4 segments as voltage sensors.Heterologous expression of channels, with mutagenesis, methane thiosulfonate reagent accessibility, and gating current experiments revealed details of the voltage-gating mechanism in sodium, potassium, and calcium channels.The identification of missense or truncation mutations in genes from patients with disorders of excitability, or channelopathies, led to their functional characterization, and expanded our understanding of the roles of diverse regions in channel function (reviewed by Cannon, 2006).The increasing number of channelopathy mutations identified and characterized as causing mixed gating defects, as well as channelopathies that promote mixed phenotypes, illustrates the challenge in the correlation of genotype to phenotype, and therefore the causality of dysfunction in channelopathy disorders.Prokaryotic sodium channels have yielded new insights into the mechanisms of channel function, with recent investigations providing detail into mechanisms of drug action and channelopathy dysfunction.Cystallographic and cryo-EM approaches have been increasingly important in the study of eukaryotic sodium channels, providing details of channel structure and enhancing computational approaches such as molecular dynamics.What has become clear is that there is no single mechanism of action for channelopathies and thus no one size fits all treatment for patients.Using diverse approaches to gain further understanding of specific genotype/phenotype relationships will facilitate more effective personalized treatment strategies that can greatly enhance patient outcomes.In this Research Topic issue, research articles on sodium channelopathies highlight advancements in our understanding of diseases of excitability, as well as the challenges inherent in bridging the gap in our knowledge of the relationship of genotype, channel dysfunction and patient phenotype.

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

How this classification was reachedexpand

Full frame machine prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. The Gemma side is a direct model label for every work in the frame, read from the title-only record. The Codex side is a classifier learned from the 10,348 direct Codex labels and calibrated to design-weighted sample rates; fields without enough sample support carry no Codex call. Candidate is the union of the two sides; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels.

metaresearch head score (Codex)0.005
metaresearch head score (Gemma)0.015
Version: metacan-v3-hybrid-931329e0061cValidation status: machine_predicted_unvalidated
Candidate categoriesnone
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Not applicable · Consensus signal: Not applicable
GenreCandidate signal: Editorial · Consensus signal: Editorial
Teacher disagreement score0.030
Threshold uncertainty score0.100

Distilled classifier scores by category (both heads)

CategoryCodexGemma
Metaresearch0.0050.015
Meta-epidemiology (narrow)0.0040.001
Meta-epidemiology (broad)0.0030.002
Bibliometrics0.0030.001
Science and technology studies0.0030.002
Scholarly communication0.0050.004
Open science0.0030.002
Research integrity0.0100.012
Insufficient payload (model declined to judge)0.0300.023

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.007
GPT teacher head0.277
Teacher spread0.270 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it

Classification

machine, unvalidated

Machine predicted; a candidate call from one source (direct Gemma or distilled Codex), not a consensus.

The models applied no category: nothing in the taxonomy fit this work.
Study designNot applicable
Domainnot available
GenreEditorial

How this classification was reached, model by model and score by score, is at the end of the page under "How this classification was reached".

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Citations0
Published2022
Admission routes1
Has abstractyes

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