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Record W4378376854 · doi:10.26434/chemrxiv-2023-1f1ct

Synthesis and ligand properties of chelating bis(N-heterocyclic carbene)-stabilized bis(phosphinidenes)

2023· preprint· en· W4378376854 on OpenAlexafffund
Jan‐Erik Siewert, Braulio M. Puerta Lombardi, N.M.H. Janssen, Roland Roesler, Christian Hering‐Junghans

Bibliographic record

VenueChemRxiv · 2023
Typepreprint
Languageen
FieldChemistry
TopicSynthesis and characterization of novel inorganic/organometallic compounds
Canadian institutionsUniversity of Calgary
FundersLeibniz-GemeinschaftLeibniz-WissenschaftsCampus Phosphorforschung RostockNatural Sciences and Engineering Research Council of CanadaMitacs
KeywordsPhosphinideneCarbeneLone pairChemistryLigand (biochemistry)DiphosphinesRhodiumMedicinal chemistryReagentAdductStereochemistryCatalysisMoleculeOrganic chemistry

Abstract

fetched live from OpenAlex

N-heterocyclic carbene-phosphinidene adducts (NHPs) are an emerging class of ligands with proven binding ability for main group and transition elements. They can be considered as inversely polarized phosphaalkenes with electron-rich P atoms possessing two lone pairs of electrons, which render them interesting platforms for the formation of multi-metallic complexes. We describe herein a modular, high-yielding synthesis of bis(NHP)s, starting from alkylidene-bridged bis(NHC)s ((IMe)}2CnH2n; n = 1,3) and a triphosphirane (cyclo-P3Dip3) (Dip = 2,6-iPr2C6H3) as phosphinidene transfer reagents. The coordination chemistry of [{DipP(IMe)}2CH2], 1, was studied in detail, and the complexes [1∙FeBr2] and [1∙Rh(cod)]Cl were prepared, showing that the ligand has a flexible bite-angle ranging between 86-106°. [1∙Rh(cod)]Cl was converted into the corresponding dicarbonyl complex [1∙Rh(CO)2]Cl, with an average value for the CO stretching frequency of 2029 cm−1, which indicates a strongly donating ligand, when compared to related bis(NHC) rhodium complexes. The binding ability of the remaining two phosphorus lone pairs was demonstrated via addition of AuCl(SMe2), which generated the hetero-trimetallic complex [1∙(AuCl)2∙Rh(cod)]Cl. Moreover, [1∙Rh(cod)]X (X− = Cl, B(3,5-CF3-C6H3)4) were tested in the catalytic hydrogenation of the α,β-unsaturated esters methyl-Z-α-acetamidocinnamate (MAC) and dimethyl itaconate (ItMe2), revealing that the chloride complex was inactive, while the BArF-complex demonstrated moderate activity, lower than that of analogous complexes incorporating classical diphosphines such as DiPAMP. In addition, [1∙Rh(cod)]Cl was shown to be moderately air- and moisture stable, slowly decomposing to the corresponding NHC-stabilized bisdioxophosphorane, which was independently synthesized by treating the free ligand with dry O2.

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

How this classification was reachedexpand

Full frame machine prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. The Gemma side is a direct model label for every work in the frame, read from the title-only record. The Codex side is a classifier learned from the 10,348 direct Codex labels and calibrated to design-weighted sample rates; fields without enough sample support carry no Codex call. Candidate is the union of the two sides; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels.

metaresearch head score (Codex)0.000
metaresearch head score (Gemma)0.000
Version: metacan-v3-hybrid-931329e0061cValidation status: machine_predicted_unvalidated
Candidate categoriesnone
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Bench or experimental · Consensus signal: Bench or experimental
GenreCandidate signal: Empirical · Consensus signal: Empirical
Teacher disagreement score0.001
Threshold uncertainty score0.003

Distilled classifier scores by category (both heads)

CategoryCodexGemma
Metaresearch0.0000.000
Meta-epidemiology (narrow)0.0000.000
Meta-epidemiology (broad)0.0000.000
Bibliometrics0.0000.000
Science and technology studies0.0000.000
Scholarly communication0.0000.000
Open science0.0000.000
Research integrity0.0000.000
Insufficient payload (model declined to judge)0.0010.000

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.051
GPT teacher head0.240
Teacher spread0.189 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it

Classification

machine, unvalidated

Machine predicted; a candidate call from one source (direct Gemma or distilled Codex), not a consensus.

The models applied no category: nothing in the taxonomy fit this work.
Study designBench or experimental
Domainnot available
GenreEmpirical

How this classification was reached, model by model and score by score, is at the end of the page under "How this classification was reached".

Quick stats

Citations0
Published2023
Admission routes2
Has abstractyes

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