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Record W4392853670 · doi:10.1136/lupus-2024-el.41

O32 Impact of patient baseline characteristics on SLE Responder Index-4 (SRI[4]) responses to deucravacitinib, a first-in-class, oral, selective, allosteric tyrosine kinase 2 inhibitor in the phase 2 PAISLEY trial in systemic lupus erythematosus

2024· article· en· W4392853670 on OpenAlex
Eric F. Morand, Cristina Arriens, Laura Geraldino‐Pardilla, Ann E. Clarke, Samantha Pomponi, Coburn Hobar, Thomas Wegman, R. Koti, Subhashis Banerjee, Ronald van Vollenhoven

Why this work is in the frame

A frame that forgets how it found something cannot be audited. These are the routes that admitted this work.

affAt least one author lists a Canadian institution in the pinned OpenAlex snapshot.

Bibliographic record

VenueOral Presentations · 2024
Typearticle
Languageen
FieldMedicine
TopicSystemic Lupus Erythematosus Research
Canadian institutionsUniversity of Calgary
FundersEMD SeronoGenentechStockholms Läns LandstingCelgeneBiogenHjärt-LungfondenGilead SciencesServierAmgenPfizerAstraZenecaEli Lilly and CompanyBristol-Myers Squibb
KeywordsAllosteric regulationIndex (typography)Tyrosine-kinase inhibitorKinaseClass (philosophy)MedicinePharmacologyChemistryInternal medicineComputer scienceReceptorBiochemistryCancerWorld Wide WebArtificial intelligence

Abstract

fetched live from OpenAlex

<h3>Objective</h3> Deucravacitinib is a first-in-class, oral, selective, allosteric tyrosine kinase 2 (TYK2) inhibitor approved in multiple countries for the treatment of adults with moderate to severe plaque psoriasis. Deucravacitinib inhibits TYK2-mediated signaling of cytokines, such as type 1 interferons, involved in systemic lupus erythematosus (SLE). In the 48-week, double-blind, phase 2 PAISLEY trial in patients with active SLE (NCT03252587), all primary and secondary endpoints were met at the 3 mg twice-daily (BID) deucravacitinib dose, including SLE Responder Index-4 (SRI[4]) response rates vs placebo at weeks 32 (primary endpoint) and 48. Week 32 response rates were 34.4% vs 58.2%, 49.5%, and 44.9% with placebo vs deucravacitinib 3 mg BID, 6 mg BID, and 12 mg once daily (QD), respectively. This exploratory analysis assessed the efficacy of deucravacitinib according to patient baseline characteristics. <h3>Methods</h3> In the PAISLEY trial, patients with active SLE were randomized 1:1:1:1 to receive placebo (n=90) or deucravacitinib 3 mg BID (n=91), 6 mg BID (n=93), or 12 mg QD (n=89). SRI(4) response rates at week 32 in the phase 2 PAISLEY trial were evaluated according to select baseline demographics and disease characteristics. Point estimates for response rates with asymptotic CIs were calculated for each treatment arm within each subgroup. All analyses were descriptive. <h3>Results</h3> SRI(4) response rates in most analyzed subgroups were consistent with the observed response rates in the overall population and favored the 3 mg BID deucravacitinib dose. SRI(4) response rates in subgroups defined by race, baseline SLEDAI-2K and glucocorticoid dose, and years since initial diagnosis are provided below (figure 1). Of these, Black/African American race, other race, baseline SLEDAI-2K of &lt;10, baseline glucocorticoid dose of ≥10 mg/day, and 3–6 and ≥6 years since diagnosis showed the greatest difference in SRI(4) responses for those receiving deucravacitinib vs placebo. <h3>Conclusion</h3> Deucravacitinib was associated with improved SRI(4) response rates at week 32 across race, SLEDAI-2K, glucocorticoid dose, and years since diagnosis at baseline subgroups. Data interpretation for some subgroups was limited by low patient numbers. These findings support the efficacy of deucravacitinib in the treatment of patients with active SLE, regardless of patient baseline characteristics. <h3>Acknowledgements</h3> We thank the patients and their families who made this study possible, as well as the clinical teams who participated. This study was sponsored by Bristol Myers Squibb. Professional medical writing assistance was provided by Angela R. Eder, PhD, of SciMentum, Inc, a Nucleus Group Holdings, Inc, company, and funded by Bristol Myers Squibb. <h3>COI Disclosures</h3> <b>EM:</b> Research support: AbbVie, Amgen, AstraZeneca, Biogen, Bristol Myers Squibb, Eli Lilly, EMD Serono, Genentech, GSK, Janssen, and UCB; Consultancy: AstraZeneca, Biogen, Bristol Myers Squibb, Eli Lilly, EMD Serono, Genentech, Gilead, Novartis, and Servier <b>CA:</b> Grant support: AstraZeneca and Bristol Myers Squibb; Advisor or review panel: AstraZeneca, Aurinia, Bristol Myers Squibb, GSK, and Kezar; Speaker/honoraria: AstraZeneca and Aurinia <b>LGP:</b> Consultancy: Aurinia and Bristol Myers Squibb <b>AC:</b> Research support: AstraZeneca and GSK; Consultancy/Speaker: AstraZeneca and GSK; Consultancy: Bristol Myers Squibb, Otsuka, and Roche <b>SP, CH, TW, and SB:</b> Employees and shareholders: Bristol Myers Squibb <b>RK:</b> Employee of Syneos Health, providing statistical services to Bristol Myers Squibb <b>RvV:</b> Research support: Bristol Myers Squibb, GSK, and Eli Lilly; Research support, consultancy, and speaker: UCB; Support for educational programs, consultancy, and speaker: Pfizer; Support for educational programs: Roche; Consultancy and speaker: AbbVie, Galapagos, and Janssen; Consultancy: AstraZeneca, Biogen, Biotest, Celgene, Gilead, and Servier

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

Full frame distilled prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. Learned from the 10,348 direct Codex labels and 10,348 direct Gemma labels. Candidate is the union of thresholded teacher heads; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels or direct frontier model labels.

metaresearch head score (Codex)0.002
metaresearch head score (Gemma)0.003
Version: codex-gemma-dda1882f352aValidation status: machine_predicted_unvalidated
Candidate categoriesMeta-epidemiology (narrow)
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Randomized trial · Consensus signal: none
GenreCandidate signal: Empirical · Consensus signal: Empirical
Teacher disagreement score0.447
Threshold uncertainty score1.000

Codex and Gemma teacher scores by category

CategoryCodexGemma
Metaresearch0.0020.003
Meta-epidemiology (narrow)0.0000.000
Meta-epidemiology (broad)0.0010.000
Bibliometrics0.0020.003
Science and technology studies0.0000.000
Scholarly communication0.0000.000
Open science0.0000.000
Research integrity0.0000.001
Insufficient payload (model declined to judge)0.0000.000

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.043
GPT teacher head0.378
Teacher spread0.335 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it