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Record W4405658272 · doi:10.1002/jsde.12826

Glucose‐induced self‐assembly in structurally diverse polyoxyethylene based nonionic surfactants for enhanced anticancer drug solubilization

2024· article· en· W4405658272 on OpenAlexaff
Ketan Kuperkar, Virendra Prajapati, D. Gerrard Marangoni, Pratap Bahadur

Bibliographic record

VenueJournal of Surfactants and Detergents · 2024
Typearticle
Languageen
FieldChemistry
TopicSurfactants and Colloidal Systems
Canadian institutionsSt. Francis Xavier University
Fundersnot available
KeywordsChemistrySolubilizationNonionic surfactantDrugCombinatorial chemistryOrganic chemistryPulmonary surfactantPharmacologyBiochemistry

Abstract

fetched live from OpenAlex

Abstract This study investigates the influence of glucose in inducing the micellar growth/transition in several structurally diverse, longer, and shorter chain polyoxyethylene (POE)‐based nonionic surfactants, commercially known as Kolliphor® HS15 (Solutol), Kolliphor EL®, Akypo®, Brij®‐78, Pluronic® (P103 and F77), Tetronic® (T1304), and Tyloxapol® in aqueous solution environment. It was observed that the addition of glucose induces dehydration of the POE moieties or chains in the tested systems, thereby enhancing the inter‐micellar interactions via hydrogen bonding in the hydrophilic part of the selected surfactants. This dehydration leads to an interesting clouding behavior across all the studied surfactant systems. Also, the dynamic light scattering (DLS) technique accounted for the probable self‐assembly and micellar growth in water and 1 M glucose ( fix ) across various temperatures. Being pharmaceutical excipients, these micellar entities were successfully employed to assay the hydrophobic anticancer drug curcumin (Cur) solubilized, as confirmed by the peak intensity variation from UV–visible spectroscopy. Cur solubilization into glucose‐containing micelles revealed enhanced solubility expressed in terms of drug loading efficiency (DL%), encapsulation efficiency (EE%), partition coefficient (log P), and standard free energy of solubilization (Δ G °), which is due to the glucose‐induced hydrophobicity in the examined nonionic micellar systems.

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

How this classification was reachedexpand

Full frame distilled prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. Learned from the 10,348 direct Codex labels and 10,348 direct Gemma labels. Candidate is the union of thresholded teacher heads; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels or direct frontier model labels.

metaresearch head score (Codex)0.001
metaresearch head score (Gemma)0.000
Version: codex-gemma-dda1882f352aValidation status: machine_predicted_unvalidated
Candidate categoriesMeta-epidemiology (narrow)
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Bench or experimental · Consensus signal: Bench or experimental
GenreCandidate signal: Empirical · Consensus signal: Empirical
Teacher disagreement score0.040
Threshold uncertainty score1.000

Codex and Gemma teacher scores by category

CategoryCodexGemma
Metaresearch0.0010.000
Meta-epidemiology (narrow)0.0000.000
Meta-epidemiology (broad)0.0010.000
Bibliometrics0.0000.000
Science and technology studies0.0000.000
Scholarly communication0.0000.001
Open science0.0000.000
Research integrity0.0000.000
Insufficient payload (model declined to judge)0.0000.000

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.015
GPT teacher head0.268
Teacher spread0.252 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it

Classification

machine, unvalidated

Machine predicted; a candidate call from one teacher head, not a consensus.

Study designBench or experimental
Domainnot available
GenreEmpirical

How this classification was reached, model by model and score by score, is at the end of the page under "How this classification was reached".

Quick stats

Citations6
Published2024
Admission routes1
Has abstractyes

Explore more

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