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Record W566310660 · doi:10.1096/fasebj.21.5.a645-b

FRET analysis of Calmodulin Binding to Nitric Oxide Synthase Peptides and Enzymes

2007· article· en· W566310660 on OpenAlexafffund
Donald E. Spratt, Valentina Taiakina, J. Guy Guillemette

Bibliographic record

VenueThe FASEB Journal · 2007
Typearticle
Languageen
FieldBiochemistry, Genetics and Molecular Biology
TopicCancer, Hypoxia, and Metabolism
Canadian institutionsUniversity of Waterloo
FundersNatural Sciences and Engineering Research Council of Canada
KeywordsCalmodulinFörster resonance energy transferChemistryCofactorNitric oxide synthaseEnzymeBiochemistryCysteineBiophysicsIsozymeAlexa FluorMutagenesisGene isoformFluorescenceMutantBiology

Abstract

fetched live from OpenAlex

Calmodulin (CaM) is a ubiquitous Ca 2+ ‐sensor protein that binds and activates the Nitric Oxide Synthase (NOS) isozymes. Although the structure of CaM has been determined when bound to a peptide derived from the CaM‐binding domain of endothelial NOS, the conformation of CaM when bound to the three mammalian NOS holoenzymes has yet to be determined. Förster Resonance Energy Transfer (FRET) is a useful method for the determination of the distance between two different fluorescently labeled residues separated by ~10 to ~100 Å. The goal of our research is to determine the conformation of CaM when bound to all three NOS isoforms through the use of FRET. We have produced a double cysteine CaM mutant (T34C/T110C) using site‐directed mutagenesis for these FRET measurements. The NOS enzymes contain three cofactors (heme, FMN, and FAD) that absorb light strongly between 250 and 500 nm. In order to avoid undesired quenching, far‐red shifted fluorescent dyes (Alexa Fluor 546 C 5 ‐maleimide and DABMI) were chosen so that they can be selectively excited in the presence of the NOS cofactors. FRET studies were performed on the fluorescently labeled CaM with stoichiometric amounts of synthetic CaM‐binding domain NOS peptides and enzymes. These studies will provide a better understanding of the inherent differences between the Ca 2+ ‐dependent and Ca 2+ ‐independent binding of CaM to the mammalian NOS isozymes. This work is supported by NSERC.

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

How this classification was reachedexpand

Full frame machine prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. The Gemma side is a direct model label for every work in the frame, read from the title-only record. The Codex side is a classifier learned from the 10,348 direct Codex labels and calibrated to design-weighted sample rates; fields without enough sample support carry no Codex call. Candidate is the union of the two sides; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels.

metaresearch head score (Codex)0.000
metaresearch head score (Gemma)0.000
Version: metacan-v3-hybrid-931329e0061cValidation status: machine_predicted_unvalidated
Candidate categoriesnone
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Bench or experimental · Consensus signal: Bench or experimental
GenreCandidate signal: Empirical · Consensus signal: Empirical
Teacher disagreement score0.001
Threshold uncertainty score0.004

Distilled classifier scores by category (both heads)

CategoryCodexGemma
Metaresearch0.0000.000
Meta-epidemiology (narrow)0.0000.000
Meta-epidemiology (broad)0.0010.000
Bibliometrics0.0000.000
Science and technology studies0.0000.000
Scholarly communication0.0000.000
Open science0.0010.000
Research integrity0.0010.001
Insufficient payload (model declined to judge)0.0010.000

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.011
GPT teacher head0.261
Teacher spread0.250 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it

Classification

machine, unvalidated

Machine predicted; a candidate call from one source (direct Gemma or distilled Codex), not a consensus.

The models applied no category: nothing in the taxonomy fit this work.
Study designBench or experimental
Domainnot available
GenreEmpirical

How this classification was reached, model by model and score by score, is at the end of the page under "How this classification was reached".

Quick stats

Citations0
Published2007
Admission routes2
Has abstractyes

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