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Record W2259435605 · doi:10.1021/ja5006724

Reactivity of Ruthenium Phosphido Species Generated through the Deprotonation of a Tripodal Phosphine Ligand and Implications for Hydrophosphination

2014· article· en· W2259435605 on OpenAlexafffund
Peter E. Sues, Alan J. Lough, Robert H. Morris

Bibliographic record

VenueJournal of the American Chemical Society · 2014
Typearticle
Languageen
FieldChemistry
TopicAsymmetric Hydrogenation and Catalysis
Canadian institutionsUniversity of Toronto
FundersNatural Sciences and Engineering Research Council of Canada
KeywordsChemistryPhosphineLigand (biochemistry)DeprotonationRutheniumMoietyMedicinal chemistryStereochemistryReactivity (psychology)CatalysisOrganic chemistry

Abstract

fetched live from OpenAlex

The fragmentation of the 1,1,2-tris(diphenylphosphino)ethane ligand in [RuCp*((Ph2P)2CHCH2PPh2)][PF6] (1) was explored through treatment with base under aprotic conditions. The neutral phosphido complex RuCp*(PPh2CH═CHPPh2)(PPh2) (2) with a (Z)-1,2-bis(diphenylphosphino)ethene (dppen) ligand was generated through a base-facilitated dehydrophosphination reaction. Installation of a bis(p-tolyl)phosphido ligand was attempted by combining bis(p-tolyl)phosphine with RuCp*(dppen)Cl in the presence of KOtBu, but surprisingly, the unsymmetrical diphenylphosphido compound RuCp*(Ph2PCHCHP(p-tol)2)(PPh2) (5) was generated instead. The ligand rearrangement reaction was driven by the greater electron density on the bis(p-tolyl)phosphido moiety. Density functional theory calculations showed that fragmentation to the 1,2-disubstituted ligand was thermodynamically favored over the 1,1-disubstituted ligand and that intramolecular phosphido exchange was kinetically accessible at room temperature. The greater basicity of the bis(p-tolyl)phosphido ligand was experimentally verified by the measured pKaTHF of 28 for the acid/base pair [RuCp*(Ph2P(o-C6H4)PPh2)(P(p-tolyl)2H)]+/RuCp*(Ph2P(o-C6H4)PPh2)(P(p-tolyl)2) versus 25 for the acid/base pair [RuCp*(Ph2P(o-C6H4)PPh2)(PPh2H)]+/RuCp*(Ph2P(o-C6H4)PPh2)(PPh2) (7). For comparison, the approximate pKaTHF values for free P(p-tolyl)2H/[K(crypt)]P(p-tolyl)2 and free PPh2H/[K(crypt)]PPh2 are 43 and 38, respectively. This is the first quantitative measurement of the large effect that coordination to a metal center, in this case ruthenium(II), has on the acidity of secondary phosphines. This is useful information for designing and understanding hydrophosphination catalysts. Complexes 2 and 7 are catalysts for the addition of PPh2H to acrylonitrile, but they deactivate fairly rapidly. The pKaTHF measurements are consistent with a catalytic cycle involving a Michael addition step. Complex 2 in solution underwent a slow, unprecedented rearrangement of P–C, C–C, and C–H bonds to give crystalline Ru(C5(CH3)4(CH2C6H5))(Ph2PCH2CH2PPh(o-C6H4)PPh) (9) in high yields, demonstrating the unpredictable reactivity of phosphido ligands.

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

How this classification was reachedexpand

Full frame distilled prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. Learned from the 10,348 direct Codex labels and 10,348 direct Gemma labels. Candidate is the union of thresholded teacher heads; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels or direct frontier model labels.

metaresearch head score (Codex)0.000
metaresearch head score (Gemma)0.001
Version: codex-gemma-dda1882f352aValidation status: machine_predicted_unvalidated
Candidate categoriesnone
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Bench or experimental · Consensus signal: Bench or experimental
GenreCandidate signal: Empirical · Consensus signal: Empirical
Teacher disagreement score0.006
Threshold uncertainty score0.277

Codex and Gemma teacher scores by category

CategoryCodexGemma
Metaresearch0.0000.001
Meta-epidemiology (narrow)0.0000.000
Meta-epidemiology (broad)0.0000.000
Bibliometrics0.0000.001
Science and technology studies0.0000.000
Scholarly communication0.0000.000
Open science0.0000.000
Research integrity0.0000.000
Insufficient payload (model declined to judge)0.0000.000

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.012
GPT teacher head0.252
Teacher spread0.241 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it

Classification

machine, unvalidated

Machine predicted; a candidate call from one teacher head, not a consensus.

The models applied no category: nothing in the taxonomy fit this work.
Study designBench or experimental
Domainnot available
GenreEmpirical

How this classification was reached, model by model and score by score, is at the end of the page under "How this classification was reached".

Quick stats

Citations35
Published2014
Admission routes2
Has abstractyes

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