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Record W4383683835 · doi:10.58931/cibdt.2023.115

JAK inhibitors for the treatment of inflammatory bowel disease

2023· article· en· W4383683835 on OpenAlex

Why this work is in the frame

A frame that forgets how it found something cannot be audited. These are the routes that admitted this work.

affAt least one author lists a Canadian institution in the pinned OpenAlex snapshot.

Bibliographic record

VenueCanadian IBD Today · 2023
Typearticle
Languageen
FieldBiochemistry, Genetics and Molecular Biology
TopicInflammatory Bowel Disease
Canadian institutionsUniversity of Calgary
Fundersnot available
KeywordsTofacitinibJanus kinaseMedicineInflammatory bowel diseaseImmunologyUlcerative colitisImmunosuppressionPsoriasisRheumatoid arthritisSTAT proteinJAK-STAT signaling pathwayTyrosine kinasePharmacologyDiseaseSignal transductionSTAT3Internal medicineCytokineBiologyReceptor

Abstract

fetched live from OpenAlex


 
 
 Over the past decade, Janus kinase (JAK) inhibitors have been developed for the treatment of several immune-mediated inflammatory diseases, including ulcerative colitis (UC) and Crohn’s disease (CD). The JAK-signal transducer and activator of transcription (STAT) pathway plays an essential role in coordinating the human immune response. Phosphorylation and activation of the JAK family of tyrosine kinases results in subsequent activation of intracytoplasmic STAT pathways with upregulation of inflammatory gene transcription. Blocking this signalling results in broad-spectrum immunosuppression, which is effective in the treatment of rheumatoid arthritis (RA), psoriasis, atopic dermatitis, and inflammatory bowel disease (IBD). To date, three oral, small-molecule JAK inhibitors (tofacitinib, filgotinib, and upadacitinib) have received regulatory approval in various jurisdictions globally for the treatment of moderate-to-severely active UC. It is anticipated that upadacitinib will soon become the first novel, advanced oral small molecule therapy approved for moderate-to-severely active CD. While these agents are highly effective, emerging data has highlighted potentially relevant safety signals associated with JAK inhibitors, and that the therapeutic index of these therapies may be distinct from that of monoclonal antibodies. Therefore, JAK inhibitors have a unique position in the therapeutic armamentarium for IBD. Here, we summarize the evidence supporting the use of JAK inhibitors and provide an overview of their practical applications in clinical care.
 
 

Fetched live from OpenAlex and de-inverted. Abstracts are not stored in this database: the inverted indexes are 8.6 GB of the frame’s 9.3 GB of text, and the host has 13 GB free.

Full frame distilled prediction

Teacher imitation

Not calibrated prevalence, not ground truth. Human validation pending. Learned from the 10,348 direct Codex labels and 10,348 direct Gemma labels. Candidate is the union of thresholded teacher heads; consensus is their intersection. These outputs are machine_predicted_unvalidated and are not human labels or direct frontier model labels.

metaresearch head score (Codex)0.000
metaresearch head score (Gemma)0.000
Version: codex-gemma-dda1882f352aValidation status: machine_predicted_unvalidated
Candidate categoriesnone
Consensus categoriesnone
DomainCandidate signal: none · Consensus signal: none
Study designCandidate signal: Not applicable · Consensus signal: Not applicable
GenreCandidate signal: Empirical · Consensus signal: Empirical
Teacher disagreement score0.139
Threshold uncertainty score0.988

Codex and Gemma teacher scores by category

CategoryCodexGemma
Metaresearch0.0000.000
Meta-epidemiology (narrow)0.0000.000
Meta-epidemiology (broad)0.0000.000
Bibliometrics0.0000.000
Science and technology studies0.0000.000
Scholarly communication0.0000.000
Open science0.0000.000
Research integrity0.0000.000
Insufficient payload (model declined to judge)0.0000.000

Machine scores (provisional)

The two teacher heads of the student model, read on this work. A score orders the frame for review; it never asserts a category, and the validation status ships verbatim with every row.

Baseline scores from an immature model (maturity gate not passed, 7 training rounds). Scores rank; they never assert a category.

Opus teacher head0.009
GPT teacher head0.227
Teacher spread0.218 · how far apart the two teachers sit on this one work
Validation statusscore_only:v0-immature-baseline · verbatim from the scoring run: score_only means the number may rank works, and no category label ships from it